| Patent # | Description |
|---|---|
| US-4,123,551 |
2,2-Disubstituted-phenylcarbamoyl-6-hydroxy-m-dioxin-4-one derivatives
having insecticidal properties Compounds of the formula I ##STR1## wherein R.sub.1 represents a phenyl group substituted by one or two members selected from the group consisting of... |
| US-4,123,550 |
Bicyclo[3.1.0]hexylethylaminocarbonyl-substituted heteroaryl
cardiovascular agents 1-Alkylamino-3-([2-(endobicyclo[3.1.0]hex-6-yl)ethylaminocarbonyl]thienylox y)-2-propanols and methods for preparing these compounds are disclosed. The compounds... |
| US-4,123,549 |
N-(3,5-dihalophenyl)-.alpha.-spirocycloalkanesuccinimides, and their
preparation and use N-(3,5-Dihalophenyl)-.alpha.-spirocycloalkanesuccinimides of the formula: ##STR1## wherein X is a chlorine or bromine atom and R is a C.sub.3 -C.sub.6 ... |
| US-4,123,548 |
(2-Oxo-pyrrolidines)-acetic hydrazides The present invention pertains to novel (2-oxo-pyrrolidine-1)-acetic hydrazides, methods for preparation and subsequent treatment therewith, and pharmaceutical... |
| US-4,123,547 |
Thienamycin sulfoxide and sulphone Thienamycin sulfoxide (I, n=1), Thienamycin sulfone (I, n=2), and their pharmaceutically acceptable salts are disclosed to be useful as antibiotics: ... |
| US-4,123,546 |
Antidepressant compounds Antidepressant compounds such as 2-[(4b,4c-dihydro-8bH-azirino[2,1,3-cd]dibenzo[a,f]pyrrolizin-8b-yl)oxy]et hyl-N,N-dimethylamine useful for alleviating... |
| US-4,123,545 |
N-Propyl-3(.beta.-hydroxyethyl)-3-(meta-hydroxyphenyl)-pyrrolidine The present invention provides a compound of the formula ##STR1## which possesses pharmacological activity, for example anti-psychotic activity. |
| US-4,123,544 |
Acetylsalicylic acid derivatives This invention relates to acetylsalicylic acid derivatives of the formula ##STR1## wherein R is H or OH, which have good analgesic, anti-inflammatory, and ... |
| US-4,123,543 |
Derivatives of substituted indoline lactans with effect on the central
nervous system New pharmacodynamically active nitrogen-containing heterocyclic compounds of the general formula ##STR1## as well as methods of preparing the same; and... |
| US-4,123,542 |
Derivatives of N-alkyl imidazoles Compounds of the formula ##STR1## wherein R is lower alkyl; R.sup.1 is substituted or unsubstituted phenyl or phenyl straight chain lower alkyl; R.sup.2 is... |
| US-4,123,541 |
2-Aminomethyl-5-phenyloxazoles and the pharmaceutically acceptable salts
thereof 2-Aminomethyl-5-phenyloxazoles and the pharmaceutically acceptacle salts thereof have been found to be effective for meliorating inflammation in warm blooded... |
| US-4,123,540 |
Isoclavulanic acid as an antibacterial and a .beta.-lactamase inhibitor .beta.-Lactamase inhibitory and antibacterial compounds of the formula: ##STR1## wherein R is a hydrogen atom or an acyl group and salts and esters thereof,... |
| US-4,123,539 |
6-Ethylpenicillanic acid Disclosed are the antibiotics 6-ethylpenicillanic acid and 6-ethylpenicillanic acid sulfoxide (I): ##STR1## Also disclosed are processes for preparing I and... |
| US-4,123,538 |
(2-Amino-2-oxoethoxy)acetic acid compounds, compositions and methods Novel (2-amino-2-oxoethoxy)acetic acid compounds and antisecretory compositions and methods employing (2-amino-2-oxoethoxy)acetic acid compounds are disclosed.... |
| US-4,123,537 |
2-Halo-4-aminomethyl-6-alkyl-3-pyridinols useful as diuretics in
treating hypertension and edema Certain substituted 4-aminomethyl-3-pyridinols and their pharmaceutically acceptacle acid addition salts wherein the pyridinol nucleus may be further substituted... |
| US-4,123,536 |
Dialkyl
({[3-(alkoxycarbonyl)-1,4-dihydro-4-oxo-8-quinolinyl]amino}methylene)pro
panedioates The present invention relates to dialkyl ({[3-(alkoxy-carbonyl)-1,4-dihydro-4-oxo-8-quinolinyl]amino}methylene)-pro panedioates having the following structural... |
| US-4,123,535 |
Psychostimulating 14-amino-14,15-dihydroeburnamenines This invention provides new compounds of formula I, ##STR1## wherein X is hydrogen or halogen having an atomic number from 9 to 35 in the 10- or... |
| US-4,123,534 |
Adenine derivatives and hypolipidemic composition thereof Adenine derivatives, their preparation and pharmaceutical compositions containing the same in an amount sufficient to effect hypolipidemia. The derivatives are... |
| US-4,123,533 |
Fused pyrimidine derivatives and compositions for treating
atherosclerosis containing them Compounds of the formula: ##STR1## or pharmaceutically acceptable salts thereof are disclosed wherein R is hydrogen or C.sub.1 to C.sub.6 alkyl; R.sup.2 and... |
| US-4,123,532 |
Method for treatment of asthma A method is provided for treatment of asthma by administering to a mammalian host a pyrazolo[1,5-c]quinazolin-5(6H)-one of the structure ##STR1## wherein... |
| US-4,123,531 |
Anti-convulsant N-ethanolamine diphenyl acetamides This invention relates to novel acetamides, the nitrogen of which is substituted with an amino lower alkyl chain. This invention also relates to a process for... |
| US-4,123,530 |
N-cyclohexyl-piperazino acetamides and propionamides New piperazine derivatives and homologs thereof of formula ##STR1## wherein n is equal to 2 or 3 and m to 1, 2 or 3; X REPRESENTS HYDROGEN OR A METHYL... |
| US-4,123,529 |
Phenylpiperazine derivatives Phenylpiperazine derivatives of formula (I): ##STR1## where R.sup.1 is benzyl, C.sub.1-6 alkyl or optionally substituted phenyl; R.sup.2 is optionally... |
| US-4,123,528 |
3-(Substituted thio) cephalosporins, derivatives and nuclear analogues
thereof Disclosed is a class of cephalosporins including the carba, aza and oxa nuclear analogues thereof which bear at the 3-position a substituted thio substituent;... |
| US-4,123,527 |
N-tricyclic derivatives of azetidine and process for their preparation Novel N-tricyclic derivatives of azetidine are disclosed of the general formula ##STR1## where A is a C.sub.1 -C.sub.3 alkylene group, a C.sub.2 -C.sub.3 ... |
| US-4,123,526 |
Thionophosphate insecticide activators Compounds which are useful as insecticide activators are described herein. The compounds are defined by the following formula: ##STR1## wherein R is... |
| US-4,123,525 |
Sublimable insecticidal compositions containing triisopropyl- or
tritertiary-butyl-s-trioxane carriers An improvement is provided in sublimable agricultural chemical compositions in the form of rough grains, pulverized powders or tablets which comprises at least... |
| US-4,123,524 |
Synthesis of
6-amino-4-methyl-8-(.beta.-D-ribofuranosyl)pyrrolo[4,3,2-de]pyrimido[4,5
... The compound 6-amino-4-methyl-8-(.beta.-D-ribofuranosyl)pyrrolo[4,3,2-de]pyrimido[4,5-c ]pyridazines-5'-phosphate (a nucleotide) as a new compound and its method ... |
| US-4,123,523 |
Analgesic and sedative polypeptides The disclosure relates to novel polypeptides which possess analgesic and sedative activity, to processes for their manufacture and to compositions containing... |
| US-4,123,522 |
Control of bloat in ruminants Bloat, particularly feedlot bloat, in ruminants is treated and controlled by the administration of the antibiotic S 15-1. This antibiotic can also be employed to... |
| US-4,123,521 |
Antibiotic U-53,946 and process for preparing the same New antiobiotic U-53,946 produced by the controlled fermentation of the new microorganism Paecilomyces abruptus sp. nov., NRRL 11110. This antibiotic is active... |
| US-4,123,520 |
Method for preparing high molecular weight meningococcal Group C vaccine A vaccine against Group C meningococcal meningitis consisting of a polysaccharide of which at least 80% by weight has a molecular weight in excess of 1,000,000... |
| US-4,123,519 |
Injectable contraceptive vaccine and method An injectable contraceptive vaccine, a method of preparing said vaccine and the method of preventing conception in mammals by use of said vaccine, is disclosed.... |
| US-4,123,518 |
Insecticidal phosphate ester-based solid composition with depot gas
action In a pesticidal preparation having a depot gas action, and comprising a phosphate ester in admixture with a solid carrier, the improvement wherein said phosphate... |
| US-4,123,517 |
Toothpaste compositions Toothpaste composition having desirable compatibility with an unlimited aluminum container, which toothpaste contains a polishing material comprising hydrate of... |
| US-4,123,516 |
Quaternary compounds having anti-microbial activity Anti-microbial quaternary ammonium compounds which include the adamantane ring system linked to the quaternary ammonium group by a hydrocarbon chain or by other... |
| US-4,123,515 |
Quaternary compounds having anti-microbial activity Anti-microbiol quaternary ammonium compounds which include the adamantane ring system linked to the quaternary ammonium group by a hydrocarbon chain or by other... |
| US-4,123,514 |
Quaternary compounds having anti-microbial activity Anti-microbial quaternary ammonium compounds which include the adamantane ring system linked to the quaternary ammonium group by a hydrocarbon chain or by other... |
| US-4,123,513 |
Quaternary compounds having anti-microbial activity Anti-microbial quaternary ammonium compounds which include the adamantane ring system linked to the quaternary ammonium group by a hydrocarbon chain or by other... |
| US-4,123,512 |
Antibacterial oral composition An antibacterial oral composition effective to promote oral hygiene containing an antibacterial antiplaque agent and an additive which reduces staining of dental... |
| US-4,123,511 |
Therapeutic copper compositions Therapeutic copper compositions are described which are adapted to be applied as from an aerosol container to areas of human skin for the treatment of muscle... |
| US-4,123,510 |
Method for the determination of gonadotropins A simple, sensitive, reliable and safe method for determining the concentration of pituitary gonadotropins is disclosed. The method involves concentration by... |
| US-4,123,509 |
Pregnancy test A simple, sensitive, reliable and safe method and device for detecting pregnancy is disclosed. The test involves concentration by ultrafiltration of a sample of... |
| US-4,123,508 |
Apparatus and method for manufacturing deuterium enriched water Deuterium-enriched water is manufactured for use as the raw material of a heavy water manufacturing plant. The enriched water is manufactured by supplying a flow... |
| US-4,123,507 |
Process for removing sulfur and NO.sub.x components from a gas stream A feed gas containing one or more components selected from the class consisting of H.sub.2 S, SO.sub.2, SO.sub.3, COS, CS.sub.2, light mercaptans, and sulfur... |
| US-4,123,506 |
Utilization of impure steam contaminated with hydrogen sulfide Certain impure streams, especially those from geothermal sources, are polluted with hydrogen sulfide, ammonia, carbon dioxide, other gases, and finely divided... |
| US-4,123,505 |
Reducing SO.sub.2 in refinery off gas Conventionally H.sub.2 S laden gases are amine scrubbed, the H.sub.2 S sprung from the amine, converted to sulfur in the Claus process and the tail gas from the... |
| US-4,123,504 |
Method of making diamonds synthetically A method of diamond synthesis, by which a reaction mixture is prepared comprising, taken in direct contact, a carbon-containing material and a combination of... |
| US-4,123,503 |
Catalysis of phosphazene cyclics to polymer, using Lewis acid compounds Thermal polymerization of (NPCl.sub.2).sub.3,4 is improved by conducting the polymerization in the presence of Lewis Acid type compounds of Al or B. |
| US-4,123,502 |
Process for the purification of gas generated in the pressure
gasification of coal A process for the purification of gas, which is generated in pressure gasification of coal, which uses a wash oil, especially tar oil, as the washing liquid to... |