| Patent # | Description |
|---|---|
| US-4,678,802 |
1-acylcarbamoyloxindole-3-carboxamides as antiinflammatory agents 1-Acylcarbamoyloxindole-3-carboxamides as antiinflammatory agents prepared by reaction of the 1-acylcarbamoyloxindole with an isocyanate in the presence of a... |
| US-4,678,801 |
Novel 2-oxopyrrolidine compounds, salts thereof process for the
preparation thereof as well as pharmaceutical... Novel 2-oxopyrrolidine compounds represented by the formula ##STR1## wherein R.sup.1 and R.sup.2 are hydrogen or alkyl group, respectively, A is alkylene... |
| US-4,678,800 |
Gamma-r-glutamoyl derivatives A compound of the formula ##STR1## wherein R.sub.1 and R.sub.6 independently represent hydroxy, C.sub.1 -C.sub.4 -alkoxy, substituted C.sub.1 -C.sub.4 -... |
| US-4,678,799 |
1,2(1,4)-dimethyl-4(2)-(2-hydroxyethyl)-5-nitro-imidazole antiprotozoal
agents with reduced mutagenicity A group of 4-substituted-5-nitroimidazoles is described, having effective antiprotozoal activity with much less mutagenicity than is shown by known ... |
| US-4,678,798 |
N-(azolylcarbamyl)-hydroxylamines and fungicides containing these
compounds N-(Azolylcarbamyl)-hydroxylamines of the formula ##STR1## where R is unsubstituted or substituted alkyl, alkenyl, alkoxyalkyl or cycloalkyl, or... |
| US-4,678,797 |
Biologically active agents containing substituted isoxazolidines Substituted isoxazolidines of the formula ##STR1## in which R.sup.1 represents optionally substituted alkyl, cycloalkyl, aralkyl, aryl or heteroaryl or... |
| US-4,678,796 |
2-alkylidene derivatives of 1,2,3,4-tetrahydropyridine-2,5-pyridine
carboxylic acid dialkyl esters useful for... Novel 2-(2-alkoxy-2-oxoethylidene)-1,2,3,4-tetrahydro-6-methyl-4-[2-(substituted )phenyl]-3,5-pyridinedicarboxylic acid dialkyl ester derivatives having ... |
| US-4,678,795 |
1-pyridylmethyl-2-nitromethylene-1,3-diazacycloalkane insecticides Novel insecticides of the formula ##STR1## in which R is a hydrogen atom or a lower alkyl group, X is a halogen atom, a lower alkyl group, a lower alkoxy group,... |
| US-4,678,794 |
N-pyridyl-substituted pyridine-2-carboxamide-1-oxides Compounds having the formula I ##STR1## and their pharamaceutically acceptable acid addition salts, wherein R.sub.1 is hydrogen or lower alkyl, A is a... |
| US-4,678,793 |
Heterocyclic compounds Novel p-[2(4,4-dimethyl-6-heterophenyl)substituted phenyl derivatives and salts thereof which are useful for combatting neoplasms and dermatoses including oral... |
| US-4,678,792 |
Quaternary 3,4-dihydro-isoquinolinium salts This invention relates to a compound of formula (I) ##STR1## wherein R.sub.1 and R.sub.2 are each independently hydrogen, C.sub.1 -C.sub.3 alkyl or C.sub.1... |
| US-4,678,791 |
6-phenyl-1,2-3,4,4a,5-6,10b-octahydrobenz(h)isoquinolines useful for
treating depression 6-Phenyl-1,2,3,4,4a,5,6,10b-octahydrobenz(h)isoquinolines having anti-depressant activity and methods for their preparation. |
| US-4,678,790 |
Certain .alpha.-benzyl-3-pyridylmethanols, N-oxides thereof and their
fungicidal use Novel pyridine, pyrazine and pyrimidine derivatives of the formula ##STR1## wherein R, R.sup.1, R.sup.2, R.sup.3 and R.sup.4 are as hereinafter set forth,... |
| US-4,678,789 |
Triazole antifungal agents Compounds of the general formula: ##STR1## wherein Ar is naphthyl, biphenylyl, phenyl or substituted phenyl; n is 0, 1 or 2; and Het is a heterocyclic group... |
| US-4,678,788 |
N-substituted 2-chloro-7-fluoro-10-piperazino-10,11-dihydrodibenzo (B,F)
thiepins and acid addition salts thereof N-substituted 2-chloro-7-fluoro-10-piperazino-10,11-dihydrodibenzo(b,f)thiepins are disclosed of the general formula I, ##STR1## in which R represents... |
| US-4,678,787 |
4H-1-benzopyran-4-ones and their sulfur containing analogs Novel 4H-1-benzopyran-4-ones and their sulfur containing analogs are disclosed which are efficacious for the treatment of psychosis including schizophrenia. |
| US-4,678,786 |
Pharmaceutical compositions having .beta.-adrenoceptor antagonist
activity employing pyridazinone derivatives This invention relates to (isopropyl and tertiary butyl-amino-2-hydroxypropoxy)phenyl-3[2H]-pyridazinones which have .beta.-adrenoceptor antagonist activity. |
| US-4,678,785 |
Thiadiazine compounds A thiadiazine compound of the formula: ##STR1## a method for preparing said compound and a pharmaceutical composition containing said compound, wherein X is... |
| US-4,678,784 |
Method for the treatment of LHRH diseases and conditions Fused tetracyclic benzodiazepines of the formula (I): ##STR1## where R.sup.1 is a cyclic amine such as 1-piperazine and R.sup.2 is H or a substituent as... |
| US-4,678,783 |
Substituted isoquinolinesulfonyl compounds An isoquinolinesulfonyl compound represented by the formula (I): ##STR1## wherein R.sup.1 : H, Cl, OH A : unsubstituted or substituted ethylene or... |
| US-4,678,782 |
3S-formamido azetidinone antibacterial agents, their preparation and use A monocyclic .beta.-lactam antibiotic having a formamido substitutent at the 3S-position, including compounds of the formula (I): ##STR1## and salts thereof... |
| US-4,678,781 |
3-substituted-aminomethyl cephalosporin derivatives A cephalosporin derivative of the formula I: ##STR1## in which X is S, O, CH.sub.2 or SO, R1 is (optionally-substituted)imidazol-2-yl or one of the C-7 acyl... |
| US-4,678,780 |
Anti-spasmodic agents having a ring in the main chain A new class of anti-spasmodic compounds having two branch chains is provided. The compounds have the general formula: ##STR1## where R, X, m, n and p are... |
| US-4,678,779 |
Weight control method A method of controlling weight in a mammal comprising administering to the mammal a weight control agent for inhibiting weight gain. The weight control agent may... |
| US-4,678,778 |
Trithiophosphonate insecticides Compounds for insecticidal control, having the formula ##STR1## in which R.sub.1 is methyl or ethyl; R.sub.2 is C.sub.3 -C.sub.5 alkyl or bromo-C.sub.4... |
| US-4,678,777 |
Pest-combating agents containing phosphorus-heterocyclic compounds An arthropodicidal composition comprising an arthropodicidally effective amount of an arthropodicidally active compound and a synergistically effective amount of... |
| US-4,678,776 |
Pyridyl-thionophosphoric acid ester useful as pesticides Pesticidally active novel 2-pyridyl-thionophosphoric acid esters of the formula ##STR1## in which R is i-propyl or sec.-butyl, X each independently is... |
| US-4,678,775 |
Method of controlling pests A method of controlling a pest which comprises bringing into contact with the pest a pest-controlling amount of an agent selected from the group consisting... |
| US-4,678,774 |
Novel synergistic compositions There are disclosed novel formulations of avermectin compounds and a substrate which demonstrate markedly enhanced insecticidal activity over that which would be... |
| US-4,678,773 |
Antitumor agent An antitumor agent of the present invention comprises, as an effective ingredient, lipoteichoic acid which is extracted from gram-positive bacterial cells. |
| US-4,678,772 |
Compositions containing glycyrrhizin There are provided compositions for the prevention and for the treatment of oral diseases based on glycyrrhizin, and a drug, and for the treatment of oral, nasal... |
| US-4,678,771 |
Adsorption layer An adsorption layer for retaining liquid or gaseous organic hydrocarbons prior to such matter reaching a sealing sheet of synthetic material. The adsorption... |
| US-4,678,770 |
Three-way catalyst for lean exhaust systems Three-way catalysts containing rhodium, rare earth oxide and platinum and/or palladium of improved durability, when subjected to exhaust gases containing excess... |
| US-4,678,769 |
Apparatus for catalyst preparation by reactive sublimation The invention relates to an apparatus for preparing tantalum halide supported catalysts which comprises a container for holding the support, a container for... |
| US-4,678,768 |
Catalyst component for polymerization of olefins A catalyst component for polymerization of olefins which is prepared by contacting a product obtained by contacting (A) a magnesium alkoxide, (B) a silicon... |
| US-4,678,767 |
Process for producing a catalyst component for polymerization of olefins A process for producing a catalyst component for polymerization of olefins which comprises contacting (a) a metal oxide with (b) an organomagnesium compound... |
| US-4,678,766 |
Enhancement of shape selectivity of zeolites A method is provided for enhancing the shape selectivity of a crystalline zeolite having a silica-to-alumina mol ratio greater than 10. The method consists of... |
| US-4,678,765 |
Catalytic cracking catalysts for high octane gasoline products Catalytic cracking catalysts, the process of their preparation and the process of their use. Cracking catalysts are disclosed for improving the octane number of... |
| US-4,678,764 |
Reactivation of noble metal-zeolite catalysts A method for reactivating noble metal-containing zeolites containing sulfur oxide poisoned noble metal such as oxygen regenerated platinum zeolite beta... |
| US-4,678,763 |
Method for reclaiming heat-damaged catalysts Heat-damaged ZSM-5 type catalysts are reclaimed by hydrothermal treatment with an aqueous medium followed by base exchange with an ammonium salt. |
| US-4,678,762 |
Very smooth and flat polycrystalline alumina substrates from direct
firing This invention provides thin, flat, water-impervious polycrystalline ceramic bodies composed of at least 99.5% by weight alumina, predominantly in the alpha... |
| US-4,678,761 |
Sinterable and strengthened magnesium oxide ceramic materials Magnesium oxide ceramic bodies may be strengthened by inclusion of zirconium oxide particles, and may be further sintered to a density approaching theoretical... |
| US-4,678,760 |
Method of forming a substantially interwoven matrix containing a
refractory hard metal and a metal compound The invention discloses an improvement in a process wherein a first reactant comprising one or more metals or metal compounds exothermically reacts with a second... |
| US-4,678,759 |
ZrB.sub.2 composite sintered material A ZrB.sub.2 composite sintered material consisting essentially of at least 1% by weight of SiC, at least 1% by weight of BN, at most 20% by weight of AlN, at... |
| US-4,678,758 |
Porous ceramic filter body and manufacturing method therefor Ceramic, porous filter body in the designed to overcome the lack of high temperature resistant thermoshock resistant and mechanical stable bodies for the... |
| US-4,678,757 |
Device and method for whole blood separation and analysis A method and device for separating blood into fluid and cellular fractions for diagnostic tests. The whole blood is introduced to a carrier containing a layer of... |
| US-4,678,756 |
Chemiluminescent sulfur detection apparatus and method In the illustrated and preferred embodiment of this disclosure, a chemiluminescent sulfur detector, both method and apparatus, for detecting bonded sulfur in... |
| US-4,678,755 |
Automatic chemical analyzer An automatic chemical analyzer performs calibration by comparing a measured value obtained by measuring a reaction solution, obtained by reacting a sample with a... |
| US-4,678,754 |
Liquid clinical control standard, and reagent products This invention relates to the field of clinical controls useful for calibrating clinical chemistry analyzers and in manual testing methods, as well as clinical... |
| US-4,678,753 |
Blood-culture flask with integrated subculture A blood-culture flask with an integrated subculture. It comprises a flask proper that can be filled with a liquid nutrient solution and has a neck with an... |