| Patent # | Description |
|---|---|
| US-5,364,896 |
Method for preparing silica filled organosiloxane compositions The triorganosiloxydiphenylsilanols of the present invention are novel silicone compounds that are useful as plasticizers for silicone rubbers. The present... |
| US-5,364,895 |
Hydrolytically stable pentaerythritol diphosphites A class of hydrolytically stable bis(aralkylphenyl)pentaerythritol diphosphites is disclosed, which is suitable as an antioxidant additives in polyolefins,... |
| US-5,364,894 |
Emulsification of asphalt and modified asphalt with primary emulsifier
polymers comprised of acrylic acid type... Emulsions of asphaltic materials, such as asphalt or asphalt blends with polymers, in water using copolymeric anionic emulsifiers are disclosed. The copolymeric... |
| US-5,364,893 |
Composition of polyepoxide and phosphorous-containing polyepoxide The invention provides epoxide resin molding compositions for protectively covering semiconductor components, which are accessible in a cost-effective manner and... |
| US-5,364,892 |
Modeling dough A modeling dough comprising gelled poly(vinyl alcohol), water and a filler provides a dough resistant to flaking, cracking, and crumbling. In the disclosed... |
| US-5,364,891 |
Incorporation of desired groups into polymers, the polymers so produced,
and compositions containing them Process for making a polymer with desired groups Y comprising reacting a precursor polymer having carbon- or nitrogen-bound --NH.sub.2 and/or --NH-- groups with... |
| US-5,364,890 |
Dental adhesive composition A compound having a carbodiimide in its molecule is incorporated in a dental adhesive composition. With this composition, dental composite material can be firmly... |
| US-5,364,889 |
Investment casting pattern material comprising thermally-collapsible
expanded microspheres A method and composition for forming investment casting patterns wherein thermally-collapsible microspheres are incorporated into the pattern composition. The... |
| US-5,364,888 |
UV light-curable epoxy-functional organopolysiloxane/polyether
composition release A UV light-curable organopolysiloxane composition which comprises (A) 100 parts by weight of an organopolysiloxane having at least one functional epoxy group in... |
| US-5,364,887 |
Process of producing methanol Methanol is catalytically produced from a synthesis gas which contains H.sub.2, CO and CO.sub.2 in a synthesis reactor at temperatures from 220.degree. to... |
| US-5,364,886 |
Process for preparing synergic antioxidant mixture An antioxidant for fat is prepared from tocopherol, ascorbic acid and lecithin. In one embodiment, a mixture of tocopherol and a lecithin first is made at a... |
| US-5,364,885 |
Reduction of hair growth Mammalian hair growth is reduced by applying to the skin a composition including pantothenic acid or an analogue of pantothenic acid. |
| US-5,364,884 |
Arginine compounds as ocular hypotensive agents The invention relates to arginine and arginine-like compounds and to methods employing these compounds as ocular hypotensive agents. These compounds are... |
| US-5,364,883 |
Isocarbocyclins for the treatment of liver and kidney diseases 16(S)-Isocarbacyclins have been found to the useful in the treatment of liver and kidney diseases. |
| US-5,364,882 |
Oxysulfonyl urea ACAT inhibitors Compounds of the formula ##STR1## wherein R is hydrogen, a straight or branched alkyl group having from 1 to 8 carbon atoms or benzyl; wherein each of... |
| US-5,364,881 |
S-alkyl-isothioureido-amino acids and use thereof Inhibitors of nitric oxide formation from arginine useful for treating hypotension, inflammation, stroke and to restore vascular contractile sensitivity to the... |
| US-5,364,880 |
Compound for treatment of cardiac arrhythmia, synthesis, and methods of
use Described is a novel compound and method, useful for treatment of cardiac arrhythmias, especially useful in patients with congestive heart failure (CHF). A... |
| US-5,364,879 |
Medical uses of trioxolane and diperoxide compounds The present invention provides a method of medical treatment for a medical condition in a mammal. In this method, a pharmacologically effective amount for... |
| US-5,364,878 |
Use of substituted 3,4-dihydro-2H-benzopyrans as remedies for
obstructive functional disorders of the lungs The use of substituted 3,4-dihydro-2H-benzopyrans as remedies for obstructive functional disorders of the lungs and/or disorders of the efferent urinary... |
| US-5,364,877 |
Indole derivatives as 5-lipoxygenase inhibitors The invention concerns a bicyclic heterocyclic derivative of the formula I ##STR1## wherein Q is an optionally substituted 9-membered bicyclic heterocyclic ... |
| US-5,364,876 |
Omega-[2-(alkyl)phenyl]-2-aminoalkanoic acids as antagonists of
excitatory amino acid receptors The present invention pertains to antagonists of excitatory amino acid receptors, their method of preparation as well as compositions pertaining to them, which... |
| US-5,364,875 |
Imidazoles linked to bicyclic heterocyclic groups for the treatment of
atherosclerosis Disclosed are imidazoles linked to bicyclic heterocyclic groups, as inhibitors of acyl-CoA:cholesterol acyltransferase (ACAT), processes for their preparation,... |
| US-5,364,874 |
Biocide composition and use A composition which contains a 2-halo-2-halomethyl glutaronitrile and a 4,5-polymethylene-4-isothiazolin-3-one. The compositions exhibit anti-microbial activity... |
| US-5,364,873 |
Pyridine-2,4- and dicarboxylic acid derivatives, the use thereof and
pharmaceutical composition based on these... The invention relates to pyridine-2,4- and -2,5-dicarboxylic acid derivatives of the formula I ##STR1## in which R.sup.1, R.sup.2 and X have the meanings... |
| US-5,364,872 |
Dihydropyridine-3,5-dicarboxylic acid ester derivatives The diastereoisomer A of a dihydropyridine-3,5-dicarboxylic acid ester derivative is provided as well as its pharmaceutically acceptable acid addition salts. The... |
| US-5,364,871 |
New thiazole derivatives, and pharmaceutical composition comprising the
same A compound of the formula: ##STR1## wherein R.sup.1 is amino, ureido, lower alkanoylamino, lower alkoxycarbonylamino, lower alkylsulfonylamino, lower ... |
| US-5,364,870 |
Fungicidal (2-aryl-2-substituted)ethyl-1,2,4-triazoles This invention relates to novel (2-aryl-2-substituted)ethyl-1,2,4- triazoles and the enantiomorphs, acid addition salts and metal salt complexes thereof, as well... |
| US-5,364,869 |
Heterocycle-substituted benzyaminopyridine angiotensin II receptor
antagonists Compounds are disclosed having the formula: ##STR1## wherein D is a substituted heterocycle, especially substituted pyridyl, E-G is a linking group,... |
| US-5,364,868 |
Amino-substituted benzoylguanidines, process for their preparation,
their use as a medicament and medicament... Amino-substituted benzoylguanidines, process for their preparation, their use as a medicament and medicament containing them Benzoylguanidines of the formula I ... |
| US-5,364,867 |
4-phenylpiperdine agents for treating cns disorders 4-Phenylpiperidines of the formula ##STR1## wherein R.sub.1 is hydrogen, hydroxy or lower-alkoxy; R.sub.2 is hydrogen, hydroxy, lower-alkanoyl, aroyl,... |
| US-5,364,866 |
Heteroarylpiperidines, pyrrolidines and piperazines and their use as
antipsychotics and analetics Heteroarylpiperidines, pyrrolidines, and piperazines are useful as antipsychotic and analgesic agents. The compounds are especially useful for treating psychoses... |
| US-5,364,865 |
Phenoxy- and phenoxyalkyl-piperidines as antiviral agents Compounds of the formula ##STR1## wherein R.sub.1 is selected from ##STR2## Y is a bond or lower alkylene; R.sub.2 and R.sub.3 are independently ... |
| US-5,364,864 |
1,4-disubstituted piperidines, their preparation and their application
in therapy 1,4-disubstituted piperidines of formula 1: ##STR1## as well as the therapeutically acceptable salts of these molecules. The invention also relates to the... |
| US-5,364,863 |
Specific 5-HT.sub.3 antagonists This invention provides bicyclic carboxylic esters and amides, their pharmaceutical formulations, and a method for their use in treating migraine, emesis,... |
| US-5,364,862 |
Compounds having antihypertensive and anti-ischemic properties This invention relates to adenosine derivatives and analogs which possess adenosine agonist activity and are useful as anti-hypertensive and anti-ischemic... |
| US-5,364,861 |
Optical isomers of
7-[3-(1,1-dialkylmethyl-1-amino-1-pyrrolidinyl]-quinolones and
naphthyridones as... Optically pure isomers of 7-[3-(1,1-dialkylmethyl-1-amino)-1-pyrrolidinyl]quinolones and naphthyridones as therapeutically active and safe antibacterial agents... |
| US-5,364,860 |
Naphthyridine compounds which inhibit tyrosine kinase and their
pharmaceutical compositions The present invention relates to the derivatives of the formula ##STR1## and their addition salts, and to their use in therapeutics, especially as drugs... |
| US-5,364,859 |
Imidazonaphthyridine derivatives Disclosed are imidazonaphthyridine derivatives represented by formula (I) ##STR1## wherein: R.sup.1 represents lower alkyl or substituted or unsubstituted ... |
| US-5,364,858 |
Camptothecin analogs as potent inhibitors of topoisomerase I A method for synthesizing camptothecin and camptothecin analogs using a novel hydroxyl-containing tricyclic intermediate and the camptothecin analogs produced by... |
| US-5,364,857 |
Combination having a neuroprotective effect The effect of neuroprotective 5-HT.sub.2 -receptorantagonistic 4-fluoro-phenyl compounds is intensified synergistically by 5-HT.sub.1A -receptoragonistic... |
| US-5,364,856 |
6-heterocyclic-4-amino-1,3,4,5-tetrahydrobenz[CD]indoles 6-heterocyclic-4-amino-1,3,4,5-tetrahydrobenz[cd]indoles are provided which are useful in modifying the function of serotonin in mammals. |
| US-5,364,855 |
4-cinnolinyl- and 4-naphthyridinyl-dihydropyridines, processes for their
preparation and their use in medicaments The invention relates to new 4-cinnolinyl- and 4-naphthyridinyl-dihydropyridines of the general formula I ##STR1## in which R.sup.1 to R.sup.5 have the... |
| US-5,364,854 |
Derivatives of substituted imidazo benzoxazin-1-one and process for
their preparation Derivatives of 2,3,3a,4-tetrahydro-2-azabicyclo alkyl-1H-imidazo[5,1,-c][1,4]benzoxazin-1-one are provided of general formula (I) ##STR1## in which... |
| US-5,364,853 |
Thioformamide derivatives Thioformamide compounds of formula (I) are disclosed in which R is alkyl, Y is methylene, ethylene or a direct bond, A is optionally substituted phenyl or... |
| US-5,364,852 |
Preparation of compact or cellular elastomers containing urethane and
urea groups, and moldings produced therefrom Compact or cellular elastomers containing urethane and urea groups are prepared by reacting a) at least one organic and/or modified organic polyisocyanate b) at least... |
| US-5,364,851 |
Conformationally restricted biologically active peptides, methods for
their production and uses thereof Electrochemical methods, preferably the Kolbe coupling reaction, are utilized to create intramolecularly bridged peptides, segments or peptide isosteres which... |
| US-5,364,850 |
Substituted tyrosyl diamide compounds The present invention provides substituted tyrosyl diamide compounds of general Formula I: ##STR1## and the pharmaceutically-acceptable salts thereof, which... |
| US-5,364,849 |
1-[3 or 4-[1-[4-piperazinyl]]-2 arylpropionyl or butryl]-heterocyclic
derivatives Piperazine derivatives of formula ##STR1## and their pharmaceutically acceptable acid addition salts are disclosed. In the formula n is 1 or 2, R is... |
| US-5,364,848 |
Substituted cephalosporin sulfones as anti-inflammatory and
antidegenerative agents New substituted cephalosporin sulfones are found to be potent elastase inhibitors and thereby useful anti-inflammatory/antidegenerative agents. |
| US-5,364,847 |
Inhibitors of sex steroid biosynthesis and methods for their production
and use Certain steroidal and non-steroidal compounds have been found to inhibit androgen and estrogen formation. Such inhibition may aid in the reduction of the... |