| Patent # | Description |
|---|---|
| US-5,466,721 |
Citral acetal ethers of alpha-hydroxy phenyl ketones and radiation
curable compositions thereof Provided are compounds having the formula: ##STR1## wherein: R.sup.1 and R.sup.2 are independently selected from the group consisting of a hydrogen atom, an... |
| US-5,466,720 |
Method of producing dimethyl ether In a method of producing dimethyl ether from a mixed gas containing carbon monoxide and either or both of hydrogen and water vapor or a mixed gas of them further... |
| US-5,466,719 |
Polyglycerol fatty acid ester mixture Polyglycerol fatty acid ester mixtures of mono- di- and polyesters of polyglycerols having a degree of polymerization of 2 to 8 and at least one saturated and/or... |
| US-5,466,718 |
Tyrosinase inhibitors Methods and compositions are provided for inhibiting the activity of tyrosinase in a host and, as a result, inhibiting melanin-formation. The ... |
| US-5,466,717 |
Halogenated 4'-methoxyacetophenones as microbicides and preservatives Halogenated 4'-methoxyacetophenones of formula I: ##STR1## wherein X is a halogen; Y is a halogen; and n is 1 or 2 as microbicides for inhibiting the growth... |
| US-5,466,716 |
Liposomal trimethylsphingosine Liposomal N,N,N-Trimethylsphingosine and pharmaceutical compositions comprising same. |
| US-5,466,715 |
3,4-disubstituted phenols-immunomodulating agents Certain 3,4-disubstituted phenols and pharmaceutically acceptable salts thereof are provided which mimic IL-1 activity by inducing IL-2 synthesis and subsequent... |
| US-5,466,714 |
Spermicidal and cytocidal fatty acid compositions This invention is directed to spermicidal or cytocidal activity of fatty acids and monoglycerides. More particularly, this invention is directed to the killing... |
| US-5,466,713 |
Iloprost with action against cerebral malaria This invention relates to the use of iloprost for the production of an agent for treating cerebral malaria. |
| US-5,466,712 |
Substituted n-aryl-1,2-diaminocyclobutene-3,4-diones The compound of the formula (I) or a pharmaceutically acceptable salt thereof, are smooth muscle relaxants ##STR1## |
| US-5,466,711 |
Medicaments A method for treating or preventing a Pneumocystis carinii infection in a mammal by administering a certain naphthoquinone compound or physiologically acceptable... |
| US-5,466,710 |
Heterobicycloalkanes as pesticidal compounds The present invention provides a class of substituted bicyclooctanes of formula ##STR1## wherein R is a C.sub.2-10 non-aromatic hydrocarbyl optionally... |
| US-5,466,709 |
Ring-substituted 2-amino-1,2,3,4-tetrahydronaphthalenes,
3-aminochromanes, and 3-aminothiochromanes The present invention provides novel ring-substituted 2-amino-1,2,3,4-tetrahydronaphthalenes, 3-aminochromanes, and 3-aminothiochromanes, including their... |
| US-5,466,708 |
Oxetanones Novel compounds of the formula ##STR1## wherein Q, R.sup.1 and R.sup.2 are described herein, are disclosed along with pharmaceutical compositions, methods... |
| US-5,466,707 |
Dimercapto-1,3-dithiolo-2-one or thione maleimides, compositions
containing them and their use as antimicrobial... Various 4,5-dimercapto-1,3-dithiolo-2-one or thione maleimides corresponding to the formula ##STR1## wherein R represents --H, phenyl, benzyl, phenethyl, a... |
| US-5,466,706 |
9H-imidazo[1,2-A]benzimidazole-3-acetamide derivatives, their
preparation and their therapeutic application Compound corresponding to the formula: ##STR1## in which X represents one or more of hydrogen, halogen, alkyl, trifluoromethyl, alkoxy, alkylthio,... |
| US-5,466,705 |
Triazole derivatives pest controlling agent and pest control method There are provided triazole derivatives represented by a general formula ##STR1## (wherein R.sup.1 is an alkyl group having a carbon number of 1-4, R.sup.2 ... |
| US-5,466,704 |
N-substituted imidazole and benzimidazole derivatives useful as
angiotenson II antagonists Compounds are disclosed having the formula ##STR1## These compounds inhibit the action of angiotensin II and are useful, therefore, for example, as... |
| US-5,466,703 |
Insecticidal and miticidal composition The invention provides an insecticidal and miticidal composition containing 2-(2,6-difluorophenyl)-4-(2-ethoxy-4-tertiarybutylphenyl)-2-oxazoline and at least... |
| US-5,466,702 |
Anti-neoplastic, anti-viral and ribonucleotide reductase activity
affecting pharmaceutical compositions and... A method for treating a human or non-human animal afflicted with malignant cells sensitive to parabactin or vibriobactin or a pharmaceutically acceptable salt or... |
| US-5,466,701 |
Saccharin derivative proteolytic enzyme inhibitors Compounds having the structural formula ##STR1## which inhibit the enzymatic activity of proteolytic enzymes, and processes for preparation thereof, method... |
| US-5,466,700 |
Anesthetic use of N-phenyl-N-(4-piperidinyl)amides The use of particular opioids to induce and maintain anesthesia and conscious sedation is disclosed. The opioids used in the method of the present invention... |
| US-5,466,699 |
Indolyl compounds for treating migraine |
| US-5,466,698 |
Substituted tetrahydrophyridines and hydroxypiperidines as central
nervous system agents Substituted tetrahydropyridines and hydroxypiperidines and derivatives thereof are described, as well as methods for the preparation and pharmaceutical... |
| US-5,466,697 |
8-phenyl-1,6-naphthyridin-5-ones The disclosed 8-aryl-1,6-naphthyridin-5-ones, compounds of Formula I, ##STR1## wherein: R.sub.1 is hydrogen, alkyl, lower alkyl, cycloalkyl, heteroalkyl, ... |
| US-5,466,696 |
Tacrine and cytochrome P450 oxidase inhibitors and methods of use Described is a method of treating Alzheimer's disease in a patient comprising administering to said patient an effective amount of tacrine in combination with a... |
| US-5,466,695 |
Method for stimulating hair growth with cationic derivative of minoxidil
using therapeutic iontophoresis This invention relates to a method of applying a cationic derivative of Minoxidil which is transported by means of iontophoresis to hair follicles where the... |
| US-5,466,694 |
Compositions for slowing down hair loss and for inducing and stimulating
its growth, based on... Composition for slowing down hair loss and inducing and stimulating its growth, comprising a compound of the following formula: ##STR1## wherein R.sub.1 and... |
| US-5,466,693 |
Granular fungicidal composition for application to an aquatic environment A fungicidal, herbicidal or plant growth regulating composition for application to an aquatic environment, the composition comprising a solid carrier, a... |
| US-5,466,692 |
Substituted pyridopyrimidines and antihypertensives This invention relates to substituted pyridopyrimidinones of general formula (I): ##STR1## wherein R.sup.1 and R.sup.2 are independently H, lower alkyl... |
| US-5,466,691 |
Thiophene compound Thiophene compounds of the formula ##STR1## wherein each symbol is as defined in the specification, their pharmaceutically acceptable salts, pharmaceutical... |
| US-5,466,690 |
Acetylenes disubstituted with a heteroaromatic group and a tetralin
group and having retinoid like activity Retinoid-like activity is exhibited by compounds of the formula ##STR1## where R is hydrogen or lower alkyl; A is pyridyl, thienyl, furyl, pyridazinyl,... |
| US-5,466,689 |
Morpholine derivatives and their use A compound represented by the formula ##STR1## wherein X is hydrogen or a substituent; R.sup.1 is an optionally substituted hydrocarbon residue; R.sup.2 and... |
| US-5,466,688 |
Pyrido[3,4-B]indole derivatives as serotonergic agents The compound of the formula: ##STR1## where R.sub.1 and R.sub.5 are independently hydrogen, fluorine, chlorine, bromine, iodine, trifluoromethyl, cyano,... |
| US-5,466,687 |
Arylidene-1-azacycloalkanes and arylalkyl-1-azacyclo-alkanes, their
salts, medicaments containing these... The invention relates to arylidene-1-azacycloalkanes and arylalkyl-1-azacycloalkanes of the general formula ##STR1## (wherein n, m, p, A, W.sup.1, W.sup.2,... |
| US-5,466,686 |
Amides of 4-oxo-azetidine-2-sulfonic acids and salts thereof, processes
for their preparation and their use The invention relates to the novel 4-oxo-azetidine-2-sulfonic acid amides and their salts of the formula I ##STR1## wherein the radicals have the meanings:... |
| US-5,466,685 |
Inhibition of expression of beta-lactamase using esters of fatty acid
alcohols A class of chemical compounds comprising fatty acid ester derivatives used to inhibit beta-lactamase production by infectious bacteria. These inhibitors have... |
| US-5,466,684 |
7-(substituted)-9-[(substituted
glycyl)amido]-6-demethyl-6-deoxytetracyclines The invention provides compounds of the formula: ##STR1## wherein R, R.sup.3, R.sup.4 and W are defined in the specification. These compounds are useful as... |
| US-5,466,683 |
Water-soluble analogs of carbamazepine The present invention relates to novel water-soluble analogs of carbamazepine and compositions containing them. The novel compositions are particularly suited... |
| US-5,466,682 |
Acylamino-alkyliden-hydroxy-bisphosphonic acids esters and salts
thereof, wherein the acyl group is derived... Compounds of formula (I) ##STR1## in which A is (CH.sub.2).sub.n in which n is 1-10, preferably 3 or 5, and R is the acyl group from a known... |
| US-5,466,681 |
Receptor conjugates for targeting penicillin antibiotics to bacteria A variety of conjugates useful for the treatment of infections due to pathogenic microorganisms are provided. The conjugates comprise at least one agent coupled... |
| US-5,466,680 |
Method and compositions for enhancing white blood cell functioning on a
mucosal or cutaneous surface The present invention relates to a method for enhancing white blood cell functioning and metabolism on a mucosal surface of a mammal. The present invention also... |
| US-5,466,679 |
Carboranyl uridines and their use in boron neutron capture therapy The invention relates to novel boron-containing nucleosides and amino acids which can utilize the enzymatic systems in tumor cells for incorporating such... |
| US-5,466,678 |
Co-administration of S-adenosyl-L-methionine to reduce the
nephrotoxicity of cisplatin therapy A pharmaceutical composition for use as a nephrotoxicity alleviator for alleviating the nephrotoxicity caused by a drug administered into the living organism,... |
| US-5,466,677 |
Dinucleoside phosphinates and their pharmaceutical compositions A dinucleotide analogue of formula ##STR1## where B.sup.1 and B.sup.2 are each independently a monovalent nucleoside base radical; R.sup.1 is R.sup.1.sub.a... |
| US-5,466,676 |
Satellite cell proliferation in adult skeletal muscle Novel methods of retroviral-mediated gene transfer for the in vivo corporation and stable expression of eukaryotic or prokaryotic foreign genes in tissues of... |
| US-5,466,675 |
Immunological activity of rhamnolipids Methods for treating various autoimmune diseases and for providing immunorestoration, by administering, to a subject in need thereof, an effective amount of a... |
| US-5,466,674 |
Bird aversion compounds A solid free flowing bird aversion compound comprising a bird aversion agent in an amount of from 10 to 80%, preferably from 30-75%, by weight of a total weight... |
| US-5,466,673 |
Method of inhibiting calcium precipitation in an intraocular irrigating
solution This invention relates to an intraocular irrigating composition containing a compound of the following formula or a pharmacologically acceptable salt thereof ... |
| US-5,466,672 |
Therapeutic use of clostridium difficile toxin A Methods for treating cancer are described, including methods for treating colon and pancreatic cancer. Bacterial toxins and portions of bacterial toxins are... |