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Patent # Description
US-5,466,721 Citral acetal ethers of alpha-hydroxy phenyl ketones and radiation curable compositions thereof
Provided are compounds having the formula: ##STR1## wherein: R.sup.1 and R.sup.2 are independently selected from the group consisting of a hydrogen atom, an...
US-5,466,720 Method of producing dimethyl ether
In a method of producing dimethyl ether from a mixed gas containing carbon monoxide and either or both of hydrogen and water vapor or a mixed gas of them further...
US-5,466,719 Polyglycerol fatty acid ester mixture
Polyglycerol fatty acid ester mixtures of mono- di- and polyesters of polyglycerols having a degree of polymerization of 2 to 8 and at least one saturated and/or...
US-5,466,718 Tyrosinase inhibitors
Methods and compositions are provided for inhibiting the activity of tyrosinase in a host and, as a result, inhibiting melanin-formation. The ...
US-5,466,717 Halogenated 4'-methoxyacetophenones as microbicides and preservatives
Halogenated 4'-methoxyacetophenones of formula I: ##STR1## wherein X is a halogen; Y is a halogen; and n is 1 or 2 as microbicides for inhibiting the growth...
US-5,466,716 Liposomal trimethylsphingosine
Liposomal N,N,N-Trimethylsphingosine and pharmaceutical compositions comprising same.
US-5,466,715 3,4-disubstituted phenols-immunomodulating agents
Certain 3,4-disubstituted phenols and pharmaceutically acceptable salts thereof are provided which mimic IL-1 activity by inducing IL-2 synthesis and subsequent...
US-5,466,714 Spermicidal and cytocidal fatty acid compositions
This invention is directed to spermicidal or cytocidal activity of fatty acids and monoglycerides. More particularly, this invention is directed to the killing...
US-5,466,713 Iloprost with action against cerebral malaria
This invention relates to the use of iloprost for the production of an agent for treating cerebral malaria.
US-5,466,712 Substituted n-aryl-1,2-diaminocyclobutene-3,4-diones
The compound of the formula (I) or a pharmaceutically acceptable salt thereof, are smooth muscle relaxants ##STR1##
US-5,466,711 Medicaments
A method for treating or preventing a Pneumocystis carinii infection in a mammal by administering a certain naphthoquinone compound or physiologically acceptable...
US-5,466,710 Heterobicycloalkanes as pesticidal compounds
The present invention provides a class of substituted bicyclooctanes of formula ##STR1## wherein R is a C.sub.2-10 non-aromatic hydrocarbyl optionally...
US-5,466,709 Ring-substituted 2-amino-1,2,3,4-tetrahydronaphthalenes, 3-aminochromanes, and 3-aminothiochromanes
The present invention provides novel ring-substituted 2-amino-1,2,3,4-tetrahydronaphthalenes, 3-aminochromanes, and 3-aminothiochromanes, including their...
US-5,466,708 Oxetanones
Novel compounds of the formula ##STR1## wherein Q, R.sup.1 and R.sup.2 are described herein, are disclosed along with pharmaceutical compositions, methods...
US-5,466,707 Dimercapto-1,3-dithiolo-2-one or thione maleimides, compositions containing them and their use as antimicrobial...
Various 4,5-dimercapto-1,3-dithiolo-2-one or thione maleimides corresponding to the formula ##STR1## wherein R represents --H, phenyl, benzyl, phenethyl, a...
US-5,466,706 9H-imidazo[1,2-A]benzimidazole-3-acetamide derivatives, their preparation and their therapeutic application
Compound corresponding to the formula: ##STR1## in which X represents one or more of hydrogen, halogen, alkyl, trifluoromethyl, alkoxy, alkylthio,...
US-5,466,705 Triazole derivatives pest controlling agent and pest control method
There are provided triazole derivatives represented by a general formula ##STR1## (wherein R.sup.1 is an alkyl group having a carbon number of 1-4, R.sup.2 ...
US-5,466,704 N-substituted imidazole and benzimidazole derivatives useful as angiotenson II antagonists
Compounds are disclosed having the formula ##STR1## These compounds inhibit the action of angiotensin II and are useful, therefore, for example, as...
US-5,466,703 Insecticidal and miticidal composition
The invention provides an insecticidal and miticidal composition containing 2-(2,6-difluorophenyl)-4-(2-ethoxy-4-tertiarybutylphenyl)-2-oxazoline and at least...
US-5,466,702 Anti-neoplastic, anti-viral and ribonucleotide reductase activity affecting pharmaceutical compositions and...
A method for treating a human or non-human animal afflicted with malignant cells sensitive to parabactin or vibriobactin or a pharmaceutically acceptable salt or...
US-5,466,701 Saccharin derivative proteolytic enzyme inhibitors
Compounds having the structural formula ##STR1## which inhibit the enzymatic activity of proteolytic enzymes, and processes for preparation thereof, method...
US-5,466,700 Anesthetic use of N-phenyl-N-(4-piperidinyl)amides
The use of particular opioids to induce and maintain anesthesia and conscious sedation is disclosed. The opioids used in the method of the present invention...
US-5,466,699 Indolyl compounds for treating migraine
US-5,466,698 Substituted tetrahydrophyridines and hydroxypiperidines as central nervous system agents
Substituted tetrahydropyridines and hydroxypiperidines and derivatives thereof are described, as well as methods for the preparation and pharmaceutical...
US-5,466,697 8-phenyl-1,6-naphthyridin-5-ones
The disclosed 8-aryl-1,6-naphthyridin-5-ones, compounds of Formula I, ##STR1## wherein: R.sub.1 is hydrogen, alkyl, lower alkyl, cycloalkyl, heteroalkyl, ...
US-5,466,696 Tacrine and cytochrome P450 oxidase inhibitors and methods of use
Described is a method of treating Alzheimer's disease in a patient comprising administering to said patient an effective amount of tacrine in combination with a...
US-5,466,695 Method for stimulating hair growth with cationic derivative of minoxidil using therapeutic iontophoresis
This invention relates to a method of applying a cationic derivative of Minoxidil which is transported by means of iontophoresis to hair follicles where the...
US-5,466,694 Compositions for slowing down hair loss and for inducing and stimulating its growth, based on...
Composition for slowing down hair loss and inducing and stimulating its growth, comprising a compound of the following formula: ##STR1## wherein R.sub.1 and...
US-5,466,693 Granular fungicidal composition for application to an aquatic environment
A fungicidal, herbicidal or plant growth regulating composition for application to an aquatic environment, the composition comprising a solid carrier, a...
US-5,466,692 Substituted pyridopyrimidines and antihypertensives
This invention relates to substituted pyridopyrimidinones of general formula (I): ##STR1## wherein R.sup.1 and R.sup.2 are independently H, lower alkyl...
US-5,466,691 Thiophene compound
Thiophene compounds of the formula ##STR1## wherein each symbol is as defined in the specification, their pharmaceutically acceptable salts, pharmaceutical...
US-5,466,690 Acetylenes disubstituted with a heteroaromatic group and a tetralin group and having retinoid like activity
Retinoid-like activity is exhibited by compounds of the formula ##STR1## where R is hydrogen or lower alkyl; A is pyridyl, thienyl, furyl, pyridazinyl,...
US-5,466,689 Morpholine derivatives and their use
A compound represented by the formula ##STR1## wherein X is hydrogen or a substituent; R.sup.1 is an optionally substituted hydrocarbon residue; R.sup.2 and...
US-5,466,688 Pyrido[3,4-B]indole derivatives as serotonergic agents
The compound of the formula: ##STR1## where R.sub.1 and R.sub.5 are independently hydrogen, fluorine, chlorine, bromine, iodine, trifluoromethyl, cyano,...
US-5,466,687 Arylidene-1-azacycloalkanes and arylalkyl-1-azacyclo-alkanes, their salts, medicaments containing these...
The invention relates to arylidene-1-azacycloalkanes and arylalkyl-1-azacycloalkanes of the general formula ##STR1## (wherein n, m, p, A, W.sup.1, W.sup.2,...
US-5,466,686 Amides of 4-oxo-azetidine-2-sulfonic acids and salts thereof, processes for their preparation and their use
The invention relates to the novel 4-oxo-azetidine-2-sulfonic acid amides and their salts of the formula I ##STR1## wherein the radicals have the meanings:...
US-5,466,685 Inhibition of expression of beta-lactamase using esters of fatty acid alcohols
A class of chemical compounds comprising fatty acid ester derivatives used to inhibit beta-lactamase production by infectious bacteria. These inhibitors have...
US-5,466,684 7-(substituted)-9-[(substituted glycyl)amido]-6-demethyl-6-deoxytetracyclines
The invention provides compounds of the formula: ##STR1## wherein R, R.sup.3, R.sup.4 and W are defined in the specification. These compounds are useful as...
US-5,466,683 Water-soluble analogs of carbamazepine
The present invention relates to novel water-soluble analogs of carbamazepine and compositions containing them. The novel compositions are particularly suited...
US-5,466,682 Acylamino-alkyliden-hydroxy-bisphosphonic acids esters and salts thereof, wherein the acyl group is derived...
Compounds of formula (I) ##STR1## in which A is (CH.sub.2).sub.n in which n is 1-10, preferably 3 or 5, and R is the acyl group from a known...
US-5,466,681 Receptor conjugates for targeting penicillin antibiotics to bacteria
A variety of conjugates useful for the treatment of infections due to pathogenic microorganisms are provided. The conjugates comprise at least one agent coupled...
US-5,466,680 Method and compositions for enhancing white blood cell functioning on a mucosal or cutaneous surface
The present invention relates to a method for enhancing white blood cell functioning and metabolism on a mucosal surface of a mammal. The present invention also...
US-5,466,679 Carboranyl uridines and their use in boron neutron capture therapy
The invention relates to novel boron-containing nucleosides and amino acids which can utilize the enzymatic systems in tumor cells for incorporating such...
US-5,466,678 Co-administration of S-adenosyl-L-methionine to reduce the nephrotoxicity of cisplatin therapy
A pharmaceutical composition for use as a nephrotoxicity alleviator for alleviating the nephrotoxicity caused by a drug administered into the living organism,...
US-5,466,677 Dinucleoside phosphinates and their pharmaceutical compositions
A dinucleotide analogue of formula ##STR1## where B.sup.1 and B.sup.2 are each independently a monovalent nucleoside base radical; R.sup.1 is R.sup.1.sub.a...
US-5,466,676 Satellite cell proliferation in adult skeletal muscle
Novel methods of retroviral-mediated gene transfer for the in vivo corporation and stable expression of eukaryotic or prokaryotic foreign genes in tissues of...
US-5,466,675 Immunological activity of rhamnolipids
Methods for treating various autoimmune diseases and for providing immunorestoration, by administering, to a subject in need thereof, an effective amount of a...
US-5,466,674 Bird aversion compounds
A solid free flowing bird aversion compound comprising a bird aversion agent in an amount of from 10 to 80%, preferably from 30-75%, by weight of a total weight...
US-5,466,673 Method of inhibiting calcium precipitation in an intraocular irrigating solution
This invention relates to an intraocular irrigating composition containing a compound of the following formula or a pharmacologically acceptable salt thereof ...
US-5,466,672 Therapeutic use of clostridium difficile toxin A
Methods for treating cancer are described, including methods for treating colon and pancreatic cancer. Bacterial toxins and portions of bacterial toxins are...
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