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Patent # Description
US-5,580,998 Process for preparing taxoids
The invention relates to a process for preparing taxoids of formula I herein that includes comprising the steps of esterifying a baccatin III derivative of the...
US-5,580,997 Baccatin III derivatives
New Baccatin III derivatives are disclosed for use in making taxoid compounds having formula (I) illustrated herein that exhibit antitumor activity.
US-5,580,996 Oxygen-containing aliphatic compounds and their use as intermediates for the preparation of 4-hydroxy-2,...
The compounds of the invention are characterised by the formulae ##STR1## wherein index p represents an integer equal to 2 or 3 and q can take the value...
US-5,580,995 Process for preparing anhydride-functional monomers
Anhydride-functional polymerizable monomers having the structure: ##STR1## and polymers and reactive compositions prepared from these monomers are ...
US-5,580,994 Preparation of tetrahydropyran-4-carboxylic acid and its esters
A process for preparing tetrahydropyran-4-carboxylic acid and its esters of the formula I ##STR1## (R=H, C.sub.1 -C.sub.8 -alkyl, C.sub.3 -C.sub.8...
US-5,580,993 Process for the preparation of iopamidol and 5-amino-2,2-dialkyl-1,3-dioxanes
A process for the preparation of Iopamidol and 5-amino-2,2-dialkyl-1,3-dioxanes of formula ##STR1## wherein R and R.sub.1 are the same or different and...
US-5,580,992 Olefinic monomers containing pendant perfluorinated cyclic ether moieties
A fluorine-containing compound represented by the following general formula (1): ##STR1## wherein A represents a group --CH.sub.2 --CH.dbd.CH.sub.2 or a...
US-5,580,991 Process for preparing butyrolactone and method for separating organic phosphorous-ruthenium complex as catalyst...
The disclosure describes a method for separating a ruthenium complex, which comprises removing an objective hydrogenation reaction product from a hydrogenation...
US-5,580,990 Pt-containing compound, process for its preparation, and application of such compounds
Pt-containing compound with the formula {Pt.sup.II (w)(x)(y)(z)} or {Pt.sup.IV (u)(v)(w)(x)(y)(z)}, wherein u, v, w, x, y and z represent whether or not the same...
US-5,580,989 Process for the preparation of N-4-[(substituted phenyl)alkylheterocyclic]- N
A process for preparing a compound of the structure I ##STR1## where A is oxygen and sulfur and R.sup.1 is selected from the group consisting of hydrogen,...
US-5,580,988 Substituted azetidines and processes of using them
New N-nitro, 3 substituted azetidine compounds are disclosed and these are sed in processes to prepare TNAZ.
US-5,580,987 Process for preparing 1-aminoacetamidopyrroles
There is disclosed a process for the preparation of 1-aminoacetamidopyrroles and 1-amino-2-(substituted)-pyrroles and related compounds of the formula ...
US-5,580,986 Substituted pyrazole derivatives
New substituted pyrazole derivatives of general formula I are described ##STR1## in which R.sup.1, R.sup.2, R.sup.3, R.sup.4, R.sup.5 and R.sup.6 have the ...
US-5,580,985 Substituted pyrazoles for the treatment of inflammation
A class of pyrazolyl compounds is described for use in treating inflammation and inflammation-related disorders. Compounds of particular interest are defined by...
US-5,580,984 Retroviral protease inhibiting compounds
A retroviral protease inhibiting compound of the formula: ##STR1## is disclosed.
US-5,580,983 Process for the preparation of N-acylated 2-chloro-5-aminomethylpyridines
2-Chloro-5-(N-acyl-aminomethyl)pyridines can be prepared by hydrogenation of 2-chloro-5-cyanopyridine with hydrogen in an acylating agent using a hydrogenation...
US-5,580,982 Substituted 3-(aminoalkylamino)-1,2-benzisoxazoles and related compounds
This application relates to compounds of the formula ##STR1## wherein R.sup.1, X, Y and n are as defined in the specification; and pharmaceutically...
US-5,580,981 Azahydroxybenzotriazoles and derivatives thereof for peptide coupling reactions
This invention relates to a process for forming an amide or an ester from a reaction between an amine or an alcohol, respectively and an acylating derivative of...
US-5,580,980 N-aminopyridone dyes
Pyridone dyes useful for thermal transfer have the formula ##STR1## wherein R.sup.1, R.sup.2, R.sup.3, Y, X and Z are defined in the specification.
US-5,580,979 Phosphotyrosine peptidomimetics for inhibiting SH2 domain interactions
The present invention makes available novel compounds represented by the general formula ##STR1## wherein Y represents a phosphate analog. Which compounds...
US-5,580,978 Process for the production of 7-ACA derivatives
The invention provides an improved process for the production of 7-amino-3-alkoxymethlycephem-4-carboxyl acid derivatives.
US-5,580,977 Process for preparing loracarbef monohydrate
The invention is directed to a crystalline anhydrate solvate of loracarbef, and also is directed to a process for preparing a crystalline monohydrate form of the...
US-5,580,976 Preparation of .beta.-lactam compounds, and intermediates therefor
A process for preparing a .beta.-lactam compound of the formula (I): ##STR1## which comprises cyclization of an azetidinone derivative of the formula: ...
US-5,580,975 Agent for keeping cut flowers fresh
An agent for keeping cut flowers fresh contains a polysaccharide gel, such as gellan gum, dispersed at a concentration of 0.05 wt. % to 1.50 wt. %, into water,...
US-5,580,974 Microfibrillated oxycellulose dispersions
Microfibrillated oxycellulose suitable for use as a carrier in agricultural, cosmetic, and topical and transdermal drug products, and as a binder and...
US-5,580,973 Process for preparing optically active nucleosides from chiral cyclobutanones
A process is disclosed for the preparation of optically active purine nucleosides, particularly nucleosides of formulae 1 and 2, nucleoside analogs and optically...
US-5,580,972 Purine nucleoside modifications by palladium catalyzed methods
This invention discloses an improved method for the preparation modified purine nucleosides at the 2-, 6-, or 8-position of the purine ring, using a palladium...
US-5,580,971 Fungal detection system based on rRNA probes
The invention includes methods for the detection of a particular genus or species of fungus in a biological sample. Some of these methods make use of a solid...
US-5,580,970 Detection of HPV transcripts
A method for detecting and/or quantitating specific DNA and/or RNA transcripts of human papillomavirus (HPV) is described. Nucleic acid probes specific for DNA...
US-5,580,969 Antisense oligonucleotides directed against human ICAM-I RNA
The present invention provides a method for the treatment of septic shock and inflammatory complications of shock. A process for selectively inhibiting the...
US-5,580,968 DNA encoding phospholipase activating protein
The invention provides methods for detecting elevated levels of phospholipase A.sub.2 activating protein in persons suspected of having rheumatoid arthritis to...
US-5,580,967 Optimized catalytic DNA-cleaving ribozymes
The present invention discloses nucleic acid enzymes capable of cleaving nucleic acid molecules, including single-stranded DNA, in a site-specific manner under...
US-5,580,966 Process for the synthesis of polyol fatty acid polyesters
The present invention pertains to a process for the production of polyol fatty acid polyesters by reacting a reactant mixture of polyol, a fatty acid lower alkyl...
US-5,580,965 Disazo dyestuffs
Disazo dyestuffs have been found which, in the form of the free acid, correspond to the formula (I) ##STR1## represents H or an optionally substituted...
US-5,580,964 Cationic thiadiazole dyestuffs
Cationic 1,3,4-thiadiazole dyestuffs of the formula ##STR1## in which the symbols used have the meaning given in the description, corresponding...
US-5,580,963 Single-chain hepatocyte growth factor variants
The invention concerns hepatocyte growth factor (HGF) variants that are resistant to proteolytic cleavage by enzymes capable of in vivo conversion of HGF into...
US-5,580,962 Parenterally administrable drug having thrombolytic activity and containing protein C
A thrombolytic, parenterally administrable drug containing activated protein C is provided for. The drug is free of serum amyloid P, thrombin activity,...
US-5,580,961 Heterodimeric T lymphocyte receptor subunit
Disclosed is a heterodimeric T lymphocyte receptor subunit. The subunit consists of variable, joining, constant, transmembrane, and cytoplasmic regions. The...
US-5,580,960 KS-laminin and methods of use
KS-laminin and a KS-laminin-kalinin adduct are disclosed. The molecules of the invention are useful for promoting the adhesion of keratinocytes to a substrate.
US-5,580,959 Purification of zein from corn gluten meal
This invention pertains to methods for extracting and purifying zein, zein bodies, glutelins or destarched corn gluten from corn gluten meal by efficiently...
US-5,580,958 Polypeptides encoding transcriptional activators and uses thereof
The invention provides a purified polypeptide having substantially the same amino acid sequence and activity as the protein having the amino acid sequence of...
US-5,580,957 GnRH analogs
Peptides which include unnatural amino acids and which either promote or inhibit the secretion of gonadotropins by the pituitary gland and inhibit the release of...
US-5,580,956 Phospholipase C-inhibiting peptides
The present invention relates to a peptide which has phospholipase C-inhibiting activity and which has the amino acid sequence defined in Sequence Listing by SEQ...
US-5,580,955 Fragments of neurofibromin (NF1) and method to reverse activated ras induced malignant transformation in...
This invention provides for a mechanism to reverse the activated Ras induced malignant transformation of mammalian cells by use of certain peptides....
US-5,580,954 Anti-obesity proteins
The present invention provides anti-obesity proteins, which when administered to a patient regulate fat tissue. Accordingly, such agents allow patients to...
US-5,580,953 Amylin antagonist peptides and uses therefor
Compounds which inhibit amylin activity are provided. These compounds may be used in the treatment of conditions where it is of benefit to reduce amylin...
US-5,580,952 Process for producing an extraction chromatography resin
A process for producing a resin for the chromatographic extraction of metal ions is provided, the process involving: treating an acidic bidentate organic phosphonate...
US-5,580,951 Method for preparing aromatic bischloroformate compositions and polycarbonates
Bischloroformate oligomer compositions are prepared by passing phosgene into a heterogeneous aqueous-organic mixture containing at least one dihydroxyaromatic...
US-5,580,950 Negative birefringent rigid rod polymer films
A class of soluble polymers having a rigid rod backbone, which when used to cast films, undergo a self-orientation process whereby the polymer backbone becomes...
US-5,580,949 Metal ion reduction in novolak resins and photoresists
The present invention provides methods for producing water insoluble, aqueous alkali soluble novolak resins having a very low level of metal ions, utilizing...
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