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Patent # Description
US-9,828,382 Pyrimidinone compounds as human neutrophil elastase inhibitors
Pyrimidone compounds defined herein exhibit human neutrophil elastase inhibitory properties and are useful for treating diseases and condition in which HNE is...
US-9,828,381 Substituted pyrazolopyrimidines and method of use
Compounds of formula (I) ##STR00001## and pharmaceutically acceptable salts thereof, wherein R.sup.1, R.sup.2, R.sup.3, R.sup.4, L.sup.1 and G.sup.1 are as...
US-9,828,380 Efficient method for the preparation of tofacitinib citrate
Disclosed is a novel process for the synthesis of tofacitinib citrate on an industrial scale with high yields and purity starting with ...
US-9,828,379 Pyrrolo-pyrrole carbamate and related organic compounds, pharmaceutical compositions, and medical uses thereof
The invention provides pyrrolo-pyrrole carbamate and related organic compounds, compositions containing such compounds, medical kits, and methods for using such...
US-9,828,378 Kinase inhibitors and methods of use
The present invention provides chemical entities or compounds and pharmaceutical compositions thereof that are capable of modulating certain protein kinases...
US-9,828,377 Heterocyclic compounds and uses thereof
Provided herein are compounds of Formula (I'') or (A''), pharmaceutical compositions comprising the compounds, and methods of use thereof. The compounds...
US-9,828,376 Substituted N-(3-pyrimidin-4-yl)phenyl)acrylamide analogs as tyrosine receptor kinase BTK inhibitors
In one aspect, the invention relates to substituted N-(3-(pyrimidin-4-yl)phenyl)acrylamide analogs, derivatives thereof, and related compounds, which are useful...
US-9,828,375 4-position substituted pyrazolopyrimidine derivative, and use thereof in drug preparation
The invention belongs to the technical field of organic synthetic drugs, and particularly relates to a pyrazolopyrimidine derivative and a preparation method...
US-9,828,374 Substituted pyrazino[2,2-a]isoquinoline derivatives
The present invention relates to compounds of formula of formula I wherein R, R.sup.1, R.sup.2 and L are as described herein, compositions containing compounds...
US-9,828,373 2-amino-pyrido[2,3-D]pyrimidin-7(8H)-one derivatives as CDK inhibitors and uses thereof
The invention provides compounds as CDK small-molecule inhibitors and uses thereof, the compounds can be used for treating inflammation and cell proliferation...
US-9,828,372 2-(1H-indazol-3-yl)-1H-imidazo[4,5-C]pyridine and therapeutic uses thereof
Indazole compounds for treating various diseases and pathologies are disclosed. More particularly, the present invention concerns the use of an indazole...
US-9,828,370 Compositions and methods for inhibiting kinases
The present invention provides compounds for the prevention or treatment of cancer or a bacterial or viral infection. Additionally, the present invention...
US-9,828,369 Isoquinoline derivatives useful as inhibitors of diacylglyceride O-acyltransferase 2
The present invention relates to a compound represented by formula I: and pharmaceutically acceptable salts thereof. The compounds of formula I are inhibitors...
US-9,828,368 Oxazole orexin receptor antagonists
The present invention is directed to oxazole compounds which are antagonists of orexin receptors. The present invention is also directed to uses of the oxazole...
US-9,828,367 Neprilysin inhibitors
In one aspect, the invention relates to compounds having the formula: ##STR00001## where R.sup.1, R.sup.2, R.sup.3, R.sup.4, and R.sup.5 are as defined in the...
US-9,828,366 Bicyclic derivatives and pharmaceutical composition including the same
The present invention relates to a novel bicyclic derivative that has an inhibitory activity against sodium-glucose linked transporters (SGLTs) present in the...
US-9,828,365 Fused tetracyclic heterocyclic compounds and methods of use thereof for the treatment of viral diseases
The present invention relates to novel Fused Tetracyclic Heterocyclic Compounds of Formula I: (I), wherein A, A', R.sup.2A, R.sup.2B, R.sup.7, R.sup.8, R.sup.9,...
US-9,828,364 Pyrazole compounds as BTK inhibitors
The present invention encompasses compounds of the formula (I) wherein the groups R.sub.1, Cy, and Y are defined herein, which are suitable for the treatment of...
US-9,828,363 Fused pyrimidines as inhibitors of P97 complex
The present invention is directed to certain fused pyrimidines having a homo or hetero cyclopentyl, cyclohexyl or cycloheptyl ring as the pyrimidine fusion...
US-9,828,362 1,4-disubstituted imidazole derivative
The present invention provides a 1,4-disubstituted imidazole derivative of formula (1') wherein ring Q.sup.1 is optionally-substituted C.sub.6-10 aryl group,...
US-9,828,361 Arylmethoxy isoindoline derivatives and compositions comprising and methods of using the same
Provided are 4'-arylmethoxy isoindoline compounds, and pharmaceutically acceptable salts, solvates, clathrates, stereoisomers, and prodrugs thereof. Methods of...
US-9,828,360 Pyrrolidinyl urea, thiourea, guanidine and cyanoguanidine compounds as TrkA kinase inhibitors
Compounds of Formula (I): or stereoisomers, tautomers, or pharmaceutically acceptable salts, or solvates or prodrugs thereof, where R.sup.1, R.sup.2, R.sup.a,...
US-9,828,359 Process for the preparation of 3-substituted (indol-1-yl)-acetic acid esters
The invention relates to an industrial scale process for the preparation of a compound of general formula (I): (Formula (I)) wherein R.sup.1, R.sup.2 and...
US-9,828,358 Compositions comprising an inhibitor of lysine specific demethylase-1
Described herein are amorphous and crystalline forms of pharmaceutically acceptable salts of the lysine specific demethylase-1 inhibitor ...
US-9,828,357 Cyclic compounds
The present invention provides compounds having a Toll-like receptor 4 (TLR4) signaling inhibitory action useful as preventive and therapeutic drugs of...
US-9,828,356 Processes and intermediates for the preparations of isomer free prostaglandis
Novel processes for the preparation of a compound of Formula I-2 substantially free of the 5,6-trans isomer: ##STR00001## wherein ##STR00002## R.sub.2,...
US-9,828,355 Compound, material for forming underlayer film for lithography, underlayer film for lithography and pattern...
The material for forming an underlayer film for lithography of the present invention contains a compound represented by the following general formula (1). ...
US-9,828,354 Biorefining compounds and organocatalytic upgrading methods
The invention provides new methods for the direct umpolung self-condensation of 5-hydroxymethylfurfural (HMF) by organocatalysis, thereby upgrading the readily...
US-9,828,352 Phenyl carbamates and their use as inhibitors of the fatty acid amide hydrolase (FAAH) enzyme and modulators of...
The invention provides compounds of Formula (I) or pharmaceutically acceptable salts thereof ##STR00001## wherein Ar', R.sub.1, R.sub.2, R.sub.3, R.sub.4,...
US-9,828,351 Enzyme interacting agents
The present disclosure relates generally, but not exclusively, to compounds and their use as enzyme interacting agents, in particular, agents which interact...
US-9,828,350 5,6-dihydro-2H-[1,4]oxazin-3-yl-amine derivatives useful as inhibitors of beta-secretase (BACE)
The present invention relates to novel 5,6-dihydro-2H-[1,4]oxazin-3-ylamine derivatives as inhibitors of beta-secretase, also known as beta-site amyloid...
US-9,828,349 1-aryl-1-hydroxy-2,3-diamino-propyl amines, 1-heteroaryl-1-hydroxy-2,3-diamino-propyl amines and related...
Compounds of the formula ##STR00001## where the variables have the meaning defined in the specification have analgesic and/or immunostimulant effect in mammals.
US-9,828,348 Benzimidazole derivatives and use thereof
The invention provides compounds that are useful as sodium channel blockers. In one aspect, the invention provides compounds of Formula I: ##STR00001## and...
US-9,828,347 Backfunctionalized imidazolinium salts and NHC carbene-metal complexes
Backfunctionalized imidazolinium salts and methods of synthesizing the same and NHC carbene-metal complexes therefrom. For backfunctionalized imidazolinium...
US-9,828,346 N-myristoyl transferase inhibitors
The present invention relates to N-heterocyclic sulphonamide compounds, in particular pyrazole sulphonamide compounds, and their use as N-myristoyl transferase...
US-9,828,345 Phenylpyrazole derivatives as potent ROCK1 and ROCK2 inhibitors
The present invention provides compounds of Formula (I): (I) or stereoisomers, tautomers, or pharmaceutically acceptable salts thereof, wherein all the...
US-9,828,344 Inhibitors of the notch signaling pathway and secretion for use in medicine
The invention relates to dihydropyridine compounds as inhibitors of the notch signalling pathway and/or inhibitors of secretion for the treatment of...
US-9,828,343 Histone demethylase inhibitors
The present invention relates generally to compositions and methods for treating cancer and neoplastic disease. Provided herein are substituted amidopyridine or...
US-9,828,342 Isatin derivatives, pharmaceutical compositions thereof, and methods of use thereof
One aspect of the invention relates to novel isatin derivative compounds and the pharmaceutical composition thereof. Another aspect of the invention relates to...
US-9,828,341 Dendritic core compounds
The invention relates to compounds that are useful for the preparation of dendrimer compounds, the use of these compounds for preparing dendrimers and processes...
US-9,828,340 Asymmetric synthesis of a substituted pyrrolidine-2-carboxamide
The invention relates to a process for the preparation of 4-{[(2R,3S,4R,5S)-3-(3-chloro-2-fluoro-phenyl)-4-(4-chloro-2-fluoro-pheny- ...
US-9,828,339 Biphenyl derivatives and methods for preparing same
Provided are biphenyl derivatives having the structure of Formula 1: ##STR00001## stereoisomers thereof, and pharmaceutically acceptable salts thereof, wherein...
US-9,828,338 Carbamate derivatives of lactam based N-acylethanolamine acid amidase (NAAA) inhibitors
Described herein are compounds and pharmaceutical compositions which inhibit N-acylethanolamine acid amidase (NAAA). Described herein are methods for...
US-9,828,337 Lysine derivative having an isothiocyanate functional group and associated method of use
A method for treating phytophotodermatitis including the steps of applying an isothiocyanate functional surfactant to an area affected by phytophotodermatitis,...
US-9,828,336 Methods and compounds useful in the synthesis of orexin-2 receptor antagonists
The present disclosure provides compounds and methods that are useful for the preparation of compounds useful as orexin-2 receptor antagonists.
US-9,828,335 Nitrone compounds and their use in personal care
Provided are compounds and compositions thereof that are useful as antioxidants in personal care formulations. The compounds are of the Formula I: ##STR00001##...
US-9,828,334 Process for preparing levomilnacipran
The present invention refers to a new process for preparing levomilnacipran, in particular to a process for the resolution of racemic tw-milnacipran with a...
US-9,828,333 Compounds for the treatment of influenza
The invention relates to oseltamivir derivatives as influenza neuraminidase inhibitors for treating influenza infections and to a method for producing said...
US-9,828,332 Non-peptide BDNF neurotrophin mimetics
Methods and compounds for treating neurological and other disorders are provided. Included is the administering to a subject in need thereof an effective amount...
US-9,828,331 Tetrahydro-isohumulone derivatives, methods of making and using
The present application provides novel tetrahydro-isohumulone (THIAA) derivatives and substantially enantiomerically pure compositions and pharmaceutical...
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