Easy To Use Patents Search & Patent Lawyer Directory

At Patents you can conduct a Patent Search, File a Patent Application, find a Patent Attorney, or search available technology through our Patent Exchange. Patents are available using simple keyword or date criteria. If you are looking to hire a patent attorney, you've come to the right place. Protect your idea and hire a patent lawyer.

Searching:





Search by keyword, patent number, inventor, assignee, city or state:




Patent # Description
US-9,834,571 Compounds for inhibiting cell proliferation in EGFR-driven cancers
The invention features compounds, pharmaceutical compositions and methods for treating patients who have an EGFR-driven cancer of Formula I: ##STR00001## ...
US-9,834,570 One step process for regioselective synthesis of .alpha.-acyloxy carbonyls
A regioselective N-Heterocyclic Carbene (NHC) catalyzed one step process for high yield synthesis of .alpha.-acyloxy carbonyl compounds is disclosed. ##STR00001##
US-9,834,569 Process for producing tetrakis(.sup.Faryl)borate salts
This invention provides processes for forming halomagnesium tetrakis(.sup.Faryl)borates, which processes comprise bringing together, in an anhydrous liquid...
US-9,834,568 Kinase inhibitors and their uses
The present disclosure provides compounds that inhibit protein kinases, such as JAK, Axl, or Syk kinases, compositions comprising the compounds and methods of...
US-9,834,567 Crystalline form of cefamandole nafate compound, preparation and preparing method thereof
A novel crystalline form is defined by diffraction angle 2.theta..degree. of X-ray powder diffraction pattern and characteristic peak of differential scanning...
US-9,834,566 Pyrazolopyrimidine macrocycles as inhibitors of human immunodeficiency virus replication
The disclosure generally relates to compounds of formula I, including compositions and methods for treating human immunodeficiency virus (HIV) infection. The...
US-9,834,565 Tricyclic heterocycles as bet protein inhibitors
The present disclosure relates to tricyclic heterocycles which are inhibitors of BET proteins such as BRD2, BRD3, BRD4, and BRD-t and are useful in the...
US-9,834,564 Substituted quinolines as PDE-10 inhibitors
Provided herein are Cyclic Nucleotide Phosphodiesterase inhibitors, and pharmaceutical compositions thereof, useful for the treatment of, for example, central...
US-9,834,563 Antidiabetic substituted heteroaryl compounds
The present invention relates to a compound represented by formula (I): and pharmaceutically acceptable salts thereof. The compounds of formula I are agonists...
US-9,834,562 7 beta-substituted 6a, 14a-ethenomorphinans and 7beta-substituted 6a, 14a-ethanomorphinans
The application is directed to a process for increasing the proportion of 7.beta.-epimer in an 7.alpha./7.beta.-epimer mixture of a 7-substituted ...
US-9,834,561 Process for preparing ibrutinib and its intermediates
The present invention provides efficient, economical, and improved methods for synthesizing ibrutinib and intermediates thereof. The invention involves a unique...
US-9,834,560 Compounds
The present invention relates to compounds of formula (I) ##STR00001## and to compositions comprising the same and to the use of the compounds and their...
US-9,834,559 4-Amino-6-phenyl-5,6-dihydroimidazo[1,5-a]pyrazin-3(2H)-one derivatives as inhibitors of beta-secretase (BACE)
The present invention relates to novel 5,6-dihydroimidazo[1,5-a]pyrazin-3(2H)-one derivatives as inhibitors of beta-secretase, also known as beta-site amyloid...
US-9,834,558 Substituted bridged urea analogs as sirtuin modulators
The present invention relates to novel substituted bridged urea compounds of Formula (I): ##STR00001## or a pharmaceutically acceptable salt thereof,...
US-9,834,557 Process for preparation of (2S, 5R)-7-oxo-6-sulphooxy-2-[((3R)-piperidine-3-carbonyl)-hydrazino ...
A process for preparation of (2S, 5R)-7-oxo-6-sulphooxy-2-[((3R)-piperidine-3-carbonyl)-hydrazino carbonyl]-1,6-diaza-bicyclo[3.2.1]octane is disclosed.
US-9,834,556 Process of preparing 3-(3-(4-aminocyclobutyl)phenyl)-5-phenyl-3H-imidazo[4,5-B]pyridin-2-YL)py- ridin-2-amine
The present invention is directed to a processes for the synthesis of 3-(3-(4-(1-aminocyclobutyl)phenyl)-5-phenyl-3H-imidazo[4,5-b]pyridin-2-yl- ...
US-9,834,555 Method for treating pain syndrome and other disorders
The present invention provides the use of certain compounds to treat peripheral or central pain syndrome and other disorders associated with the T-type calcium...
US-9,834,554 BTK inhibitors
The present invention provides Bruton's Tyrosine Kinase (Btk) inhibitor compounds according to Formula I or pharmaceutically acceptable salts thereof. Formula I...
US-9,834,553 Tetrahydroimidazopyridine derivatives as modulators of TNF activity
A series of substituted 4,5,6,7-tetrahydro-3H-imidazo[4,5-c]pyridine derivatives of formula (I), being potent modulators of human TNFa activity, are accordingly...
US-9,834,552 Inhibitor compounds
The present invention relates to compounds of formula I ##STR00001## wherein R.sub.1, R.sub.4, Ar, W, X and Z are all as defined herein. The compounds of the...
US-9,834,551 Substituted pyrrolo[2,3-b]pyrazines and substituted pyrazolo[3,4-b]pyridines as ITK and JAK kinase inhibitors
The present invention relates to compounds described by Formula I: ##STR00001## salts thereof, their synthesis, and their use as ITK and JAK3 inhibitors...
US-9,834,550 Pyridopyrimidinone compounds for modulating the catalytic activity of histone lysine demethylases (KDMs)
The present invention provides a compound of Formula (I) being capable of modulating the activity of histone lysine demethylase (KDM), pharmaceutical...
US-9,834,549 3,3-disubstituted-(8-aza-bicyclo[3.2.1]OCT-8-yl)-[5-(1H-pyrazol-4-yl)-thio- phen-3-yl]-methanones as inhibitors...
The present invention pertains generally to the field of therapeutic compounds. More specifically the present invention pertains to certain ...
US-9,834,548 Pyridazine compounds as JAK inhibitors
In one aspect, the invention provides a compound according to formula I, as well as tautomers, pharmaceutically acceptable salts, and hydrates thereof....
US-9,834,547 Molecules having certain pesticidal utilities, and intermediates, compositions, and processes related thereto
This disclosure relates to the field of molecules having pesticidal utility against pests in phyla Nematoda, Arthropoda, and/or Mollusca, processes to produce...
US-9,834,546 Insecticidal compounds
The invention relates to compounds of formula (I): ##STR00001## where A.sup.1, A.sup.2, A.sup.3, A.sup.4, G, R.sup.1, R.sup.2, R.sup.3 and R.sup.4 are as...
US-9,834,545 Modulators of chemokine receptors
Compounds are provided as chemokine inhibitors having the structure: ##STR00001##
US-9,834,544 Sweet flavor modifier
The present invention includes compounds having structural formula (I), or salts or solvates thereof. These compounds are useful as sweet flavor modifiers. The...
US-9,834,543 Indazoles and use thereof
In one aspect, the present disclosure provides indazoles of Formula I: (I) and the pharmaceutically acceptable salts and solvates thereof, wherein R.sup.3,...
US-9,834,542 LXR modulators
The present invention provides compounds of Formula I: and pharmaceutically acceptable salts or solvates thereof, as modulators of liver X receptors (LXR),...
US-9,834,541 2-aminopyridine compounds
The invention provides novel substituted 2-aminopyridine compounds according to Formula (I), their manufacture and use for the treatment of hyperproliferative...
US-9,834,540 Omeprazole Sodium semihydrate and preparation method thereof
It discloses Omeprazole Sodium semihydrate and preparation method thereof, wherein every mole of Omeprazole Sodium semihydrate contains 0.5 mole of water, and...
US-9,834,539 Pyridin-2(1H)-one quinolinone derivatives as mutant-isocitrate dehydrogenase inhibitors
The invention relates to inhibitors of mutant isocitrate dehydrogenase (mt-IDH) proteins with neomorphic activity useful in the treatment of cell-proliferation...
US-9,834,538 6-, 7-, or 8-substituted quinazolinone derivatives and compositions comprising and methods of using the same
Provided herein are quinazolinone compounds of formula (I), and pharmaceutically acceptable salts, solvates, clathrates, stereoisomers, and prodrugs thereof....
US-9,834,537 Compounds as chloride channel blocking agent
Disclosed is a novel compound to function as a calcium-dependent chloride channel blocking agent.
US-9,834,536 Method for producing catalyst for cyclic carbonate synthesis
A method for producing a heterogeneous catalyst for use of synthesizing cyclic carbonates by reacting an epoxide and carbon dioxide in the presence of the...
US-9,834,535 Sulfamate derivative compounds for use in treating or alleviating pain
The present invention relates to sulfamate derivative compounds and a composition for treating and/or alleviating pain containing the sulfamate derivative...
US-9,834,534 Neuraminidase inhibitor compounds, compositions and methods for the use thereof in anti-viral treatments
Compounds having a structure of Formula I and compositions comprising these compounds are provided. Uses of such compounds and compositions are provided for...
US-9,834,533 Process for preparing SGLT2 inhibitors and intermediates thereof
The present invention provides processes for preparing SGLT2 inhibitors, such as dapagliflozin and empagliflozin.
US-9,834,532 Stat3 pathway inhibitors and cancer stem cell inhibitors
The present invention relates to a novel naphtho class of compounds as Stat3 pathway inhibitors and as cancer stem cell inhibitors; to methods of using such...
US-9,834,531 Use of carboxylic acids and furanic molecules for esterification
A process for recovering and using an organic/carboxylic acid or furanic molecule by means of making an ester of a free carboxylic acid or furanic molecule with...
US-9,834,530 3-furyl-2-cyano-2-acrylamide derivative, preparation method therefor, pharmaceutical composition and use thereof
Disclosed are a 3-furyl-2-cyano-2-acrylamide derivative with epidermal growth factor receptor (EGFR) inhibitory activity and pharmaceutical acceptable salt...
US-9,834,529 Synthesis of benzothiazepines
Methods for preparing the following compound are disclosed. ##STR00001##
US-9,834,528 Alpha-amino esters of hydroxypropylthiazolidine carboxamide derivative and salt form, crystal polymorph thereof
The invention provides .alpha.-amino esters of a hydroxypropylthiazolidine carboxamide derivative, ...
US-9,834,527 Macrocyclic urea derivatives as inhibitors of TAFIa, their preparation and their use as pharmaceuticals
The present invention relates to macrocydic urea derivatives of the formula I (I) in which R1, R2, R3, V and Y are as defined below. The compounds of the...
US-9,834,526 HIV protease inhibitors
The present invention is directed to 2,5,6-substituted morpholine derivatives and their use in the inhibition of HIV protease, the inhibition of HIV...
US-9,834,525 Inhibitors of paxillin function and related compositions and methods
This disclosure relates to small molecule inhibitors of paxillin and paxillin binding, and related compositions and methods of treatment.
US-9,834,524 Isoxazoles, a process for their preparation and uses thereof
The present invention relates to novel isoxazoles, a process for their preparation and their use in the preparation of technical textiles and PPE's (Personal...
US-9,834,523 Method for preparing 3-trifluoromethyl chalcones
Disclosed is a method for preparing a compound of Formula 1 wherein Q and Z are as defined in the disclosure comprising distilling water from a mixture...
US-9,834,522 Multi-functional acrylates
Disclosed herein are derivatives of phenolic and melamine compounds, methods of making these derivatives, and methods of using them. The compounds include...
← Previous | 1 2 3 4 5 6 7 8 9 10 11 12 13 14 15 16 17 18 19 20 21 22 23 24 25 26 27 28 29 30 31 32 33 34 35 36 37 38 39 40 41 42 43 44 45 46 47 48 49 50 51 52 53 54 55 56 57 58 59 60 61 62 63 64 65 66 67 68 69 70 71 72 73 74 75 76 77 78 79 80 81 82 83 84 85 86 87 88 89 | Next →

File A Patent Application

  • Protect your idea -- Don't let someone else file first. Learn more.

  • 3 Easy Steps -- Complete Form, application Review, and File. See our process.

  • Attorney Review -- Have your application reviewed by a Patent Attorney. See what's included.