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Patent # Description
US-9,840,519 Macrocyclic compounds as TRK kinase inhibitors
Compounds of Formula I: and pharmaceutically acceptable salts thereof, wherein ring A, ring B, W, m, D, R.sup.2, R.sup.2a, R.sup.3, R.sup.3a, and Z are as...
US-9,840,518 MCL-1 inhibitors and methods of use thereof
Disclosed is a compound which is 17-chloro-5,13,14,22-tetramethyl-28-oxa-2,9-dithia-5,6,12,13,22-pentaazah- ...
US-9,840,517 Compound inhibiting activities of BTK and/or JAK3 kinases
The present invention relates to a compound inhibiting the activities of Bruton's tyrosine kinase (BTK) and/or Janus kinase 3 (JAK3), a pharmaceutical...
US-9,840,516 Substituted quinazolines as inhibitors of KRAS G12C
Compounds having activity as inhibitors of G12C mutant KRAS protein are provided. The compounds have the following structure (I): ##STR00001## or a...
US-9,840,515 Protein kinase D inhibitors
Compounds according to Formula (I), are potent inhibitors of protein kinase D (pan-PKD) activity. PKD controls key signaling cascades in cells, affecting cell...
US-9,840,514 Dianhydrides, polyimides, methods of making each, and methods of use
Embodiments of the present disclosure provide for an aromatic dianhydride, a method of making an aromatic dianhydride, an aromatic dianhydride-based polyimide,...
US-9,840,513 Substituted tricyclics and method of use
The present invention provides for compounds of formula (I) ##STR00001## wherein X, Y, and R.sup.1 have any of the values defined in the specification, and...
US-9,840,512 Antidiabetic bicyclic compounds
Novel compounds of the structural formula (I), and the pharmaceutically acceptable salts thereof, are agonists of G-protein coupled receptor 40 (GPR40) and may...
US-9,840,511 2-(aryl or heteroaryl-)phenyl (AZA)benzofuran compounds for the treatment of hepatitis C
Compounds of Formula I, including their salts, as well as compositions and methods of using the compounds are set forth. The compounds have activity against...
US-9,840,510 Pyrazolo[1,5-a]pyrimidinyl carboxamide compounds and their use in the treatment of medical disorders
The invention provides substituted pyrazolo[1,5-a]pyrimidinyl carboxamide and related organic compounds, compositions containing such compounds, medical kits,...
US-9,840,509 Heterocyclic compounds
The present invention relates to heterocyclic compounds of the general formula (I) their pharmaceutically acceptable salts, pharmaceutically acceptable...
US-9,840,508 N-acyl-(3-substituted)-(8-methyl)-5,6-dihydro-[1,2,4]triazolo[4,3-a] pyrazines as selective NK-3 receptor...
Novel compounds of Formula I ##STR00001## and their use in therapeutic treatments.
US-9,840,507 5,6-dihydro-imidazo[1,2-a]pyrazin-8-ylamine derivatives useful as inhibitors of beta-secretase (BACE)
The present invention relates to novel 5,6-dihydro-imidazo[1,2-a]pyrazin-8-ylamine inhibitors of beta-secretase, having the structure shown in Formula (I) ...
US-9,840,506 Crystal of doripenem, and preparation method therefor
This invention relates to a novel doripenem crystal, a solvate thereof, and a preparation method thereof and, more specifically, to a novel doripenem anhydride...
US-9,840,505 Solid forms of (S)-3-(1-(9H-purin-6-ylamino)ethyl)-8-chloro-2-phenylisoquinolin-1 (2H)-one and methods of...
Polymorphs of chemical compounds that modulate kinase activity, including PI3 kinase activity, and compounds, pharmaceutical compositions, and methods of...
US-9,840,504 Pyrazolopyridine derivatives and their use in therapy
The present invention relates to pyrazolopyridine derivatives, which are useful as medicaments, pharmaceutical compositions comprising one or more of the...
US-9,840,503 Heterocyclic compounds and uses thereof
The present disclosure relates to heterocyclic compounds, and pharmaceutical compositions of the same, that are inhibitors of the TAM protein kinases and are...
US-9,840,502 Salts and crystalline forms of an apoptosis-inducing agent
Salts and crystalline forms of 4-(4-{[2-(4-chlorophenyl)-4,4-dimethylcyclohex-1-en-1-yl]methyl}piperazin- ...
US-9,840,501 Morpholin-pyridine derivatives
The present invention relates to compounds of formula of formula I wherein X, R, L, Ar, R.sup.1 and n are as described herein, compositions containing compounds...
US-9,840,500 Compounds as dual inhibitors of histone methyltransferases and DNA methyltransferases
It relates to the use of compounds of formula (I'), or their pharmaceutically or veterinary acceptable salts, or their stereoisomers or mixtures thereof, as...
US-9,840,499 Solid forms of 3-(6-(1-(2,2-difluorobenzo[d][1,3]dioxol-5-yl)cyclopropanecarboxamido)-3-- ...
The present invention relates to a substantially crystalline and free solid state form of 3-(6-(1-(2,2-difluorobenzo[d][1,3]dioxol-5-yl) ...
US-9,840,498 Substituted quinazolin-4-one derivatives
Provided are substituted quinazolin-4-one compounds of the formula (I) and/or pharmaceutically acceptable salts and/or solvates thereof, wherein R.sup.1,...
US-9,840,497 P2X4 receptor antagonist
The present invention relates to a compound represented by the following general formula (II), wherein, in the formula, R.sup.1a to R.sup.6a represent hydrogen...
US-9,840,496 CD38 inhibitors and methods of treatment
Compounds of Formula I and methods of treating diseases of metabolism by modulating cellular NAD+ levels through the inhibition of the CD38 enzyme, are...
US-9,840,495 Oxindole derivatives carrying a piperidyl-substituted azetidinyl substituent and use thereof for treating...
The present invention relates to novel substituted oxindole derivatives of formula (I) wherein the variables are as defined in the claims and description; to...
US-9,840,494 Quinazoline derivative
Disclosed are N-[4-(3-chloro-4-fluorophenylamino)-7-(2-methoxyethoxy) quinazolin-6-yl]-2 -[1-(2-methoxyethyl)piperidin-4-ylidene]acetamide and a...
US-9,840,493 Modified amino acids comprising tetrazine functional groups, methods of preparation, and methods of their use
Provided herein are modified amino acids comprising a tetrazine groups according to Formula I: polypeptides, antibodies, payloads and conjugates comprising...
US-9,840,492 Antifungal compounds and processes for making
The present invention relates to polymorphic forms of compound 1 or 1a and processes for preparing compound 1 and 1a polymorphs, which are useful as antifungal...
US-9,840,491 Quinazolinones and azaquinazolinones as ubiquitin-specific protease 7 inhibitors
The present disclosure relates to inhibitors of USP7 inhibitors useful in the treatment of cancers, neurodegenerative diseases, immunological disorders,...
US-9,840,490 Process for the preparation of 3-(3-chloro-1H-pyrazol-1-yl)pyridine
3-(3-Chloro-1H-pyrazol-1-yl)pyridine is prepared by cyclizing 3-hydrazinopyridine-dihydrochloride with commercially available 3-ethoxyacrylonitrile to provide...
US-9,840,489 Piperidine carboxamide compound, preparation method, and usage thereof
The present invention provides a compound of a general formula I, a stereomeride, pharmaceutically acceptable salt or a solvate thereof, a preparation method...
US-9,840,488 Carbon monoxide releasing molecules and associated methods
The present disclosure relates to carbon monoxide releasing molecules ("CORMs"), and methods of synthesizing and applying the molecules. More specifically, this...
US-9,840,487 Catalytic enantioselective synthesis of 2-aryl chromenes and related phosphoramidite ligands and catalyst compounds
Methods to access 2-aryl chromene compounds via an asymmetric catalytic process.
US-9,840,486 Methods of producing alkylfurans
Provided herein are methods of producing dialkylfurans, such as 2,5-dimethylfuran, and other alkyl furans, such as 2-methylfuran. For example, 2,5-dimethylfuran...
US-9,840,485 Bisfuran dihalide, method for producing bisfuran dihalide, and method for producing bisfuran diacid, bisfuran...
A bisfuran dihalide having a structure represented by the following formula (1): ##STR00001## wherein R.sup.1 is a divalent hydrocarbon group represented by...
US-9,840,484 Aryl compound and making method
An aryl compound terminated with at least three glycidyl groups and at least three (meth)allyl groups, having formula (1) wherein R.sup.1 is a C.sub.3-C.sub.20...
US-9,840,483 Radiomitigating pharmaceutical formulations
The present disclosure relates to compounds of Formula (I) and (II), compositions containing the compounds (alone or in combination with other agents), and...
US-9,840,482 Sulfonamide derivatives and pharmaceutical applications thereof
Provided herein are sulfonamide derivatives or a stereoisomer, a geometric isomer, a tautomer, an N-oxide, a hydrate, a solvate, a metabolite, a...
US-9,840,481 Allosteric modulators of nicotinic acetylcholine receptors
The present disclosure relates to compounds of formula I that are useful as modulators of .alpha.7 nAChR, compositions comprising such compounds, and the use of...
US-9,840,480 Humic acid derivatives and methods of preparation and use
Disclosed are antioxidative natural compounds, their salts, chelates and cleavage derivatives that exhibit a superior combination of properties. The compounds...
US-9,840,479 Polyamine-fatty acid derived lipidoids and uses thereof
The present disclosure provides polyamine-fatty acid derived lipidoids (e.g., compounds of Formula (I) or (II)) and methods of preparing the lipidoids. A...
US-9,840,478 Piperazine derivatives as HIV protease inhibitors
The present invention is directed to piperazine derivatives, pharmaceutical compositions comprising the same, and their use in the inhibition of HIV protease,...
US-9,840,477 Cyclopropanecarboxamido-substituted aromatic compounds as anti-tumor agents
The present disclosure relates to novel cyclopropanecarboxamido-substituted aromatic compounds that inhibit protein kinases and their use in anti-tumor area. In...
US-9,840,476 5-fluoro-4-imino-3-(alkyl/substituted alkyl)-1-(arylsulfonyl)-3,4-dihydropyrimidin-2(1H)-one and processes for ...
Provided herein are 5-fluoro-4-imino-3-(alkyl/substituted alkyl)-1-(arylsulfonyl)3,4-dihydropyrimidin-2(1H)-one and processes for their preparation which may...
US-9,840,475 N-(substituted)-5-fluoro-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidine-1(2H- )-carboxamide derivatives
This present disclosure is related to the field of to N-(substituted)-5-fluoro-4-imino-3-methyl-2-oxo-3,4-di-hydropyrimidme-1(2- H)-carboxamide compounds and...
US-9,840,474 Pyrimidine compounds and use as anti-cervical cancer thereof
Provided is use of a pyrimidine compound or a pharmaceutically acceptable salt thereof in preparation of an anti-cervical cancer medicament. Research of the...
US-9,840,473 Method of preparing a high purity imidazolium salt
The present invention encompasses a novel method for synthesizing highly pure salts of the general formula Q.sup.+A.sup.-, wherein Q.sup.+ is: ##STR00001## and...
US-9,840,472 Compositions and methods for the treatment of mucositis
The invention relates to the compounds of formula I, formula II, formula III and formula IV or its pharmaceutical acceptable polymorphs, solvates, enantiomers,...
US-9,840,471 Compounds useful as modulators of TRPM8
The present invention includes compounds useful as modulators of TRPM8, such as compounds of Formulae (Ia), (Ib) and (Ic), and the subgenus and species thereof;...
US-9,840,470 Targeting GLI proteins in human cancer by small molecules
The present disclosure provides compositions, pharmaceutical preparations and methods for the diagnosis and treatment of cancers expressing a GLI polypeptide....
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