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Patent # Description
US-1,002,3588 Compositions and methods for treating cancer
K-Ras is the most frequently mutated oncogene in human cancer. Disclosed herein are compositions and methods for modulating K-Ras and treating cancer.
US-1,002,3587 Oxabicycloheptanes and oxabicycloheptenes, their preparation and use
This invention provides compounds having the structure ##STR00001## which may be used for the treatment of tumors.
US-1,002,3586 Enhanced regio-selectivity in glycol acylation
A method for acid-catalyzed acylation of an isohexide is described. The method involves a reaction of an isohexide and an excess of carboxylic acid in the...
US-1,002,3585 Photochromic compounds and intermediate compounds for production thereof
The invention covers new bicyclic bridged [1,3]oksazepine derivatives of the general formula (I) and (II): ##STR00001## which exhibit enhanced photochromic...
US-1,002,3584 Tetrandrine family pharmaceutical formulations and method
Drug formulations, methods and their use in treatment of diseases using formulations of pure di-acid salts of tetrandrine family members, especially...
US-1,002,3583 Bicyclic pyridine compound
The problem to be solved by the present invention is to provide a compound suitable for a pharmaceutical composition, specifically a pharmaceutically...
US-1,002,3582 6-aryl amino pyridone formamide compound crystal and preparation method therefor
The present invention provides a crystal of 6-arylamino pyridone carboxamide compound and a preparation method thereof. The crystal is obtained by dissolving ...
US-1,002,3581 Modified cytotoxins and their therapeutic use
The present disclosure generally provides compounds useful for treating cancer. In some aspects, the disclosure provides small-molecule cytotoxins that are...
US-1,002,3579 Pyrrolopyrimidine compounds, use as inhibitors of the kinase LRRK2, and methods for preparation thereof
The present disclosure is concerned with certain pyrrolopyrimidine compounds that are capable of inhibiting certain protein kinases, and especially the...
US-1,002,3578 Crystals of dispiropyrrolidine derivatives
Crystals of a dispiropyrrolidine compound or a salt thereof which inhibits the action of Mdm2 are provided. The present invention provides crystals of ...
US-1,002,3577 Crystalline form of JAK kinase inhibitor bisulfate and a preparation method thereof
A crystal form of JAK kinase inhibitor bisulfate and a preparation method thereof are provided. In particular, a type II crystal of ...
US-1,002,3576 Heteroaryl substituted pyrrolotriazine amine compounds as PI3K inhibitors
Disclosed are compounds of Formula (I); or a salt thereof; wherein Qi is (i) Cl, Br, I, --CN, --CH.sub.3, or --CF.sub.3; or (ii) pyrazole, triazole, or...
US-1,002,3575 Cyclic ether derivatives of pyrazolo[1,5-a]pyrimidine-3-carboxyamide
The invention relates to Spirocyclic ether derivatives of pyrazolo[1,5-a]pyrimidine-3-carboxyamide of general formula (I) which are inhibitors of...
US-1,002,3574 8-[3-amino-piperidin-1-yl]-xanthines, the preparation thereof and their use as pharmaceutical compositions
The present invention relates to substituted xanthines of general formula ##STR00001## wherein R.sup.1 to R.sup.3 are as defined herein, the tautomers, the...
US-1,002,3573 Beta-lactamase inhibitor and process for preparing the same
A process for preparing a diazabicyclooctane compound represented by the following formula (I): ##STR00001## wherein A represents RcO--; B represents NH or...
US-1,002,3572 2-(1h-indazol-3-yl)-3h-imidazo[4,5-b]pyridine and therapeutic uses thereof
Indazole compounds for treating various diseases and pathologies are disclosed. More particularly, the present invention concerns the use of an indazole...
US-1,002,3571 TYK2 inhibitors and uses thereof
The present invention provides compounds of formula I, ##STR00001## compositions thereof, and methods of using the same for the inhibition of TYK2, and the...
US-1,002,3570 Substituted pyrazolo[1,5-A]pyridine compounds as RET kinase inhibitors
Provided herein are compounds of the General Formula I: ##STR00001## and stereoisomers and pharmaceutically acceptable salts or solvates thereof, in which A,...
US-1,002,3569 Methods of preparing inhibitors of influenza viruses replication
A method of preparing Compound (1) or a pharmaceutically acceptable salt thereof: ##STR00001## comprises: (a) reacting Compound (X): ##STR00002## or a...
US-1,002,3568 Naphthyridine derivatives useful as .alpha..sub.v.beta..sub.6 integrin antagonists
A compound of formula (I) or a salt thereof ##STR00001## wherein R.sub.1 represents a hydrogen atom, a methyl group or a ethyl group R.sub.2 represents a...
US-1,002,3567 Imidazole and thiazole compositions for modifying biological signaling
Compounds having General Formula (I) or General Formula (II): in which R.sup.1 is chosen from C.sub.1 to C.sub.10 aliphatic or heteroaliphatic groups,...
US-1,002,3566 Dasatinib salts
The invention relates to normal or acidic salts of dasatinib and the hydrate and solvate forms thereof. More specifically the invention concerns: dasatinib...
US-1,002,3565 N,N' substituted piperidinamine compounds, and preparation method and usage thereof
The present invention relates to a compound of formula (I), a stereomeride, pharmaceutically acceptable salt, a solvate or an N-oxide thereof, a medicine...
US-1,002,3564 G protein-coupled receptor kinase 2 inhibitors and methods for use of the same
Disclosed herein are novel GRK2 inhibitors and methods for their use in treating or preventing heart disease, such as cardiac failure, cardiac hypertrophy, and...
US-1,002,3563 Cyclic compounds substituted by a condensed ring system
Compounds of formula I ##STR00001## defined herein are provided. Uses of these compounds for controlling invertebrate pests, protecting plant propagation...
US-1,002,3562 Heteroaryl substituted pyridyl compounds useful as kinase modulators
Compounds having the following formula: ##STR00001## or a stereoisomer or a pharmaceutically-acceptable salt thereof, wherein R.sup.2 is a monocyclic...
US-1,002,3561 Fumagillol heterocyclic compounds and methods of making and using same
Disclosed herein, in part, are fumagillol compounds and methods of use in treating medical disorders, such as obesity. Pharmaceutical compositions and methods...
US-1,002,3560 Crystalline salt form of (S)-(2-(6 chloro-7-methyl-1H-benzo[d]imidazol-2-yl)-2-methylpyrrolidin-1-yl)(5-meth- ...
The invention relates to a crystalline form of (S)-(2-(6-chloro-7-methyl-1H-benzo[d]imidazol-2-yl)-2-methylpyrrolidin-1-- ...
US-1,002,3559 Substituted azetidine derivatives
The present invention relates to compounds of formula of formula I wherein R, R.sup.1. R.sup.2, R.sup.2', R.sup.3, R.sup.4, R.sup.5, L.sup.1, L.sup.2 and N are...
US-1,002,3558 Compounds
Compounds of formula (I) defined herein exhibit human neutrophil elastase inhibitory properties and are useful for the treatment of disease or conditions in...
US-1,002,3557 Therapeutic inhibitory compounds
Provided herein are heterocyclic derivative compounds and pharmaceutical compositions comprising said compounds that are useful for inhibiting plasma...
US-1,002,3556 Androgen receptor modulators and uses thereof
Described herein are compounds that are androgen receptor modulators. Also described are pharmaceutical compositions and medicaments that include the compounds...
US-1,002,3555 NSAIDs derivatives and uses thereof
The present invention discloses novel compounds derived from NSAIDs and pharmaceutically acceptable salts thereof. Other aspects of the invention relate to use...
US-1,002,3554 Halogen-substituted heterocyclic compound salt
The invention provides a novel .alpha.-halogen-substituted thiophene compound salt that has a potent LPA receptor antagonistic action and is useful as a...
US-1,002,3553 Method and device for manufacturing lactide
A method and a device for manufacturing lactide, whereby crude lactide, being prepared by means of depolymerization of lactic acid oligomers, is purified by...
US-1,002,3552 Method of preparing a liquiritigenin precursor
[Problem] To provide a process suitable for mass-producing of iso-liquiritigenin. [Solution] A process for preparing iso-liquiritigenin, which comprises steps...
US-1,002,3551 Glutathione-cleavable prodrug and methods of use thereof
A glutathione-cleavable prodrug is provided herein, as well as methods for its use in treating cancer, including triple negative breast cancer. The prodrug can...
US-1,002,3550 Production of 2-substituted 4-hydroxy-4-methyltetrahydropyrans having stable odoriferous quality
The present invention relates to a method for the production of 2-substituted 4-hydroxy-4-methyltetrahydropyrans from the acid-catalyzed reaction of...
US-1,002,3549 Process for the production of 1,4-butanediol and tetrahydrofuran from furan
The present invention provides a process for the preparation of 1,4-butanediol and tetrahydrofuran said process comprising contacting furan with hydrogen and...
US-1,002,3548 Energy efficient manufacturing process for preparing N,O-triglycidyl aminophenols
The invention relates to an improved process for making monomeric triglycidyl compounds, wherein the triglycidyl compounds include N, O-triglycidyl compounds...
US-1,002,3547 Multifunctional primary amine, process for its preparation, and use thereof
The invention relates to a hydrophilically modified multifunctional amine AC which has more than one primary amino group per molecule, and at least one group...
US-1,002,3546 Acesulfame potassium compositions and processes for producing same
Improved processes for producing high purity acesulfame potassium. In one embodiment, the process comprises the steps of contacting a solvent, e.g.,...
US-1,002,3544 Heterocyclic compound
A fused heterocyclic compound having an enteropeptidase inhibitory action and use of the compound as a medicament for treatment or prophylaxis of obesity,...
US-1,002,3543 Inhibitors of lysine specific demethylase-1
The present invention relates generally to compositions and methods for treating cancer and neoplastic disease. Provided herein are substituted heterocyclic...
US-1,002,3542 Ibrutinib intermediate compounds, preparation methods and uses thereof
The present invention relates to the technical field of ibrutinib, particularly to the technical field of ibrutinib intermediate compounds and preparation...
US-1,002,3541 Urea compounds and their use as enzyme inhibitors
A compound having the following structure: ##STR00001## or a pharmaceutically acceptable salt or derivative thereof. The compound may be used in the treatment...
US-1,002,3540 Hydrogen barrier agent, hydrogen barrier film forming composition, hydrogen barrier film, method for producing...
To provide a hydrogen barrier agent capable of imparting hydrogen barrier performance to various materials; a hydrogen barrier film forming composition...
US-1,002,3539 Aryl-cyanoguanidine compounds
The present invention relates to protein-lysine N-methyltransferase SMYD2 (SET and MYND domain-containing protein 2) inhibitors, in particular SMYD2-inhibitory...
US-1,002,3538 Compounds, compositions and associated methods comprising 3-aryl quinolines
Compounds, compositions and methods useful for treating infectious diseases are provided. In particular, 3-aryl quinoline compounds, their synthesis,...
US-1,002,3537 Heterocyclic compounds for the treatment of neurological and psychological disorders
Lactam compounds of Formula I and their use for the treatment of neurological and psychiatric disorders including schizophrenia, bipolar disorder, anxiety...
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